SCHEMBL7009897

SCHEMBL7009897

COc1ccc(Cl)c(Oc2c(C=O)nc(N3CCOCC3)nc2N(CC(C)C)S(=O)(=O)c2ccccc2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 1/20 0.43
PIK3CA P42336 5/20 0.38
MTOR P42345 2/20 0.38
MAPT P10636 6/20 0.37
RORC P51449 2/20 0.36
ALDH1A1 P00352 4/20 0.36
LMNA P02545 2/20 0.36
HPGD P15428 1/20 0.36
OPRK1 P41145 1/20 0.36
PIK3CD O00329 3/20 0.36
PIK3CB P42338 2/20 0.36
KMT2A Q03164 2/20 0.35
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
GAA P10253 1/20 0.35
TSHR P16473 1/20 0.35
HTT P42858 1/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
TNF P01375 1/20 0.35
NOD2 Q9HC29 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7013707 0.91 EDNRA (0.45) EDNRAPIK3CAMTORMAPTRORC
SCHEMBL7013473 0.89 EDNRA (0.44) EDNRAPIK3CAMTORMAPTRORC
SCHEMBL7012433 0.89 EDNRA (0.47) EDNRAPIK3CAMTORMAPTRORC
SCHEMBL7018075 0.85 EDNRA (0.48) EDNRAPIK3CAMTORMAPTRORC
SCHEMBL7006907 0.83 EDNRA (0.42) EDNRAPIK3CAMTORMAPTRORC
SCHEMBL7009200 0.81 EDNRB (0.38) EDNRAMAPTRORCALDH1A1HPGD
SCHEMBL8325013 0.80 EDNRB (0.43) EDNRAPIK3CAMTORRORCEP300
SCHEMBL7293953 0.77 MCL1 (0.40) MAPTRORCALDH1A1HPGDKMT2A
SCHEMBL7850722 0.76 EDNRA (0.46) EDNRAPIK3CAMAPTALDH1A1HPGD
SCHEMBL7332509 0.75 RORC (0.38) MAPTRORCALDH1A1HPGDKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0601386-B1 Sulphonamides HOFFMANN LA ROCHE (CH) 2003-02-05 EP claimed
EP-0601386-A1 Sulphonamides F. HOFFMANN-LA ROCHE AG (CH) 1994-06-15 EP claimed
EP-0601386-B1 Sulphonamides HOFFMANN LA ROCHE (CH) 2003-02-05 EP disclosed
EP-0601386-A1 Sulphonamides F. HOFFMANN-LA ROCHE AG (CH) 1994-06-15 EP disclosed