SCHEMBL7007555

SCHEMBL7007555

CCCCOc1c2cc(Cl)c(Cl)c(=O)c-2cn(C(C)C)c1N(C)C(=O)O

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
FFAR4 Q5NUL3 1/20 0.34
THRA P10827 5/20 0.33
THRB P10828 5/20 0.33
ESR1 P03372 1/20 0.32
RXRA P19793 1/20 0.30
KDM4E B2RXH2 1/20 0.30
SLC6A5 Q9Y345 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7006211 0.86 THRA (0.32) THRATHRBESR1
SCHEMBL7006238 0.81 THRB (0.31) THRATHRB
SCHEMBL7010259 0.80 ESR1 (0.39) FFAR4THRATHRBESR1
SCHEMBL7592050 0.73 THRA (0.36) THRATHRB
SCHEMBL7006368 0.72 PTGS1 (0.32)
SCHEMBL5234729 0.72 THRB (0.36) FFAR4THRATHRBESR1KDM4E
SCHEMBL7003687 0.69 ESR1 (0.37) THRBESR1RXRA
SCHEMBL5235017 0.69 THRA (0.34) THRATHRBKDM4E
SCHEMBL7562047 0.68 TNF (0.37) ESR1
SCHEMBL5234473 0.68 THRB (0.37) THRATHRBESR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1355886-A1 FUSED HETEROCYCLIC COMPOUNDS Takeda Chemical Industries, Ltd. (JP) 2003-10-29 EP disclosed
WO-2002062764-A1 FUSED HETEROCYCLIC COMPOUNDS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-08-15 WO disclosed