Bromide

Bromide

SCHEMBL7008173

Br.CC(C)(C)NCC(=O)c1ccc(-c2ccccc2)cc1

nearest known ligand 0.56

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.56
MAPT P10636 4/20 0.56
L3MBTL1 Q9Y468 2/20 0.56
HPGD P15428 1/20 0.53
ERCC5 P28715 1/20 0.53
FEN1 P39748 1/20 0.53
HAO1 Q9UJM8 1/20 0.53
ALDH1A1 P00352 3/20 0.51
KDM4E B2RXH2 3/20 0.51
PTPN1 P18031 1/20 0.51
GSK3B P49841 1/20 0.51
USP2 O75604 1/20 0.51
RAB9A P51151 3/20 0.50
FFAR1 O14842 1/20 0.50
LMNA P02545 1/20 0.50
CYP1A2 P05177 1/20 0.50
HIF1A Q16665 1/20 0.50
AGTR1 P30556 1/20 0.49
NPC1 O15118 2/20 0.45
GAA P10253 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7006232 0.97 SMN1; SMN2 (0.56) SMN1; SMN2MAPTL3MBTL1HPGDERCC5
SCHEMBL10788888 0.88 KMT2A (0.56) SMN1; SMN2MAPTL3MBTL1HPGDERCC5
Hydrochloric Acid SCHEMBL28169360 0.86 KMT2A (0.54) SMN1; SMN2MAPTL3MBTL1HPGDERCC5
SCHEMBL6871371 0.81 ERCC5 (0.58) SMN1; SMN2HPGDERCC5FEN1ALDH1A1
Hydrochloric Acid SCHEMBL6866018 0.80 ERCC5 (0.56) SMN1; SMN2HPGDERCC5FEN1ALDH1A1
Hydrochloric Acid SCHEMBL7006229 0.80 HPGD (0.51) SMN1; SMN2MAPTL3MBTL1HPGDHAO1
SCHEMBL28309572 0.79 ALDH1A1 (0.47) SMN1; SMN2MAPTHPGDERCC5FEN1
SCHEMBL2298691 0.77 PLOD2 (0.53) SMN1; SMN2MAPTHPGDALDH1A1KDM4E
Hydrochloric Acid SCHEMBL6463561 0.77 ADRB2 (0.49) L3MBTL1ALDH1A1KDM4EPTPN1RAB9A
SCHEMBL2295669 0.77 GSK3B (0.52) MAPTHPGDHAO1ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0970084-B1 PYRROLO 2,3D]PYRIMIDINES AND THEIR USE AS TYROSINE KINASE INHIBITORS BASF AG (DE) 2003-06-04 EP disclosed
US-6001839-A Substituted 4-amino-7H-pyrrolo [2,3,-d]-pyrimidines as PTK inhibitors BASF AKTIENGESELLSCHAFT (DE) 1999-12-14 US disclosed