SCHEMBL7008487

SCHEMBL7008487

O=CCC1CNc2cc(OCCC3CCCCN3)c(C(F)(F)F)cc21

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.36
HTR2A P28223 2/20 0.33
CYP1A2 P05177 2/20 0.33
CYP2D6 P10635 2/20 0.33
LMNA P02545 2/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
TSHR P16473 1/20 0.33
CYP2C19 P33261 1/20 0.33
CACNA1F O60840 1/20 0.33
KCNA5 P22460 1/20 0.33
SLC6A2 P23975 1/20 0.33
ADRA1A P35348 1/20 0.33
OPRK1 P41145 1/20 0.33
CACNA1D Q01668 1/20 0.33
KCNH2 Q12809 1/20 0.33
CACNA1S Q13698 1/20 0.33
CACNA1C Q13936 1/20 0.33
SCN5A Q14524 1/20 0.33
LTA4H P09960 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7003860 0.85 CHEK2 (0.33) CHEK2SSTR2HSP90AA1HSP90AB1
SCHEMBL7009169 0.85 CHEK2 (0.33) HPGDCHEK2SSTR2HSP90AA1HSP90AB1
SCHEMBL7002160 0.85 HSP90AA1 (0.34) CHEK2SSTR2HSP90AA1HSP90AB1
SCHEMBL7007474 0.84 CHEK2 (0.34) CHEK2SSTR2HSP90AA1HSP90AB1
SCHEMBL7011908 0.81 CHEK2 (0.39) LTA4HCHEK2SSTR2
SCHEMBL5260910 0.70 LTA4H (0.41) HPGDCYP1A2CYP2D6LMNACYP3A4
SCHEMBL11457902 0.69 PIM1 (0.45) LTA4H
SCHEMBL5261782 0.67 PRKCZ (0.37) HTR2ALTA4H
SCHEMBL11448820 0.66 CHRNB4 (0.47) LTA4H
Hydrochloric Acid SCHEMBL11447408 0.64 LTA4H (0.50) LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1309551-A1 INDOLINE DERIVATIVES AS 5HT2C ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 2003-05-14 EP disclosed
WO-2002014273-A1 INDOLINE DERIVATIVES AS 5HT2C ANTAGONISTS SMITHKLINE BEECHAM P.L.C. (GB) 2002-02-21 WO disclosed