SCHEMBL7003860

SCHEMBL7003860

O=CCC1CNc2cc(OCCC3CCCCN3)c(I)cc21

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 1/20 0.33
SSTR2 P30874 2/20 0.32
KMT2A Q03164 1/20 0.31
HSP90AA1 P07900 1/20 0.31
HSP90AB1 P08238 1/20 0.31
PIM1 P11309 1/20 0.31
PIM2 Q9P1W9 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7009169 0.88 CHEK2 (0.33) CHEK2SSTR2KMT2AHSP90AA1HSP90AB1
SCHEMBL7002160 0.87 HSP90AA1 (0.34) CHEK2SSTR2HSP90AA1HSP90AB1
SCHEMBL7007474 0.86 CHEK2 (0.34) CHEK2SSTR2KMT2AHSP90AA1HSP90AB1
SCHEMBL7008487 0.85 HPGD (0.36) CHEK2SSTR2HSP90AA1HSP90AB1
SCHEMBL7011908 0.84 CHEK2 (0.39) CHEK2SSTR2KMT2A
SCHEMBL3580473 0.64 LTA4H (0.48) CHEK2
SCHEMBL15594561 0.63
SCHEMBL6903897 0.63
SCHEMBL7007537 0.63 ALDH1A1 (0.36) CHEK2SSTR2HSP90AA1HSP90AB1PIM1
Hydrochloric Acid SCHEMBL7323126 0.63 LTA4H (0.48) CHEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1309551-A1 INDOLINE DERIVATIVES AS 5HT2C ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 2003-05-14 EP disclosed
WO-2002014273-A1 INDOLINE DERIVATIVES AS 5HT2C ANTAGONISTS SMITHKLINE BEECHAM P.L.C. (GB) 2002-02-21 WO disclosed