SCHEMBL7008719

SCHEMBL7008719

Nc1cc(-n2cc(C(=O)O)c(=O)c3c(N)c(F)c(F)c(F)c32)c(F)cc1F

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
STAT3 P40763 2/20 0.52
ALDH1A1 P00352 2/20 0.51
HTT P42858 2/20 0.51
TOP1 P11387 5/20 0.43
TOP2A P11388 4/20 0.39
TOP2B Q02880 1/20 0.39
GSK3B P49841 6/20 0.39
POLB P06746 2/20 0.39
KDM4E B2RXH2 1/20 0.39
HSP90AA1 P07900 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
CACNA1F O60840 1/20 0.38
MAPK1 P28482 1/20 0.38
CACNA1D Q01668 1/20 0.38
KCNH2 Q12809 1/20 0.38
CACNA1S Q13698 1/20 0.38
CACNA1C Q13936 1/20 0.38
FOXO1 Q12778 1/20 0.35
SLC2A1 P11166 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6581471 0.90 TOP2A (0.42) STAT3ALDH1A1HTTTOP1TOP2A
SCHEMBL7006109 0.90 TOP1 (0.41) STAT3ALDH1A1HTTTOP1TOP2A
SCHEMBL7007135 0.89 STAT3 (0.54) STAT3ALDH1A1HTTTOP1TOP2A
SCHEMBL5868683 0.85 ALDH1A1 (0.53) STAT3ALDH1A1HTTTOP1TOP2A
SCHEMBL7010194 0.83 CACNA1F (0.51) STAT3TOP1TOP2ATOP2BGSK3B
SCHEMBL6576283 0.82 TOP1 (0.43) STAT3ALDH1A1HTTTOP1TOP2A
SCHEMBL7009597 0.82 GSK3B (0.44) STAT3ALDH1A1HTTTOP1TOP2A
SCHEMBL7009143 0.82 TOP1 (0.57) STAT3ALDH1A1HTTTOP1TOP2A
SCHEMBL8478277 0.80 TOP2A (0.53) ALDH1A1TOP1TOP2ATOP2BPOLB
SCHEMBL7011332 0.80 TOP2A (0.53) ALDH1A1TOP1TOP2ATOP2BPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0787720-B1 PYRIDONECARBOXYLATE DERIVATIVE OR SALT THEREOF AND ANTIBACTERIAL CONTAINING THE SAME AS ACTIVE INGREDIENT WAKUNAGA SEIYAKU KK (JP) 2003-07-16 EP disclosed
US-5910498-A NOVEL COMPOUNDS HAVING REDUCED CYTOTOXICITY, PHOTOTOXICITY; TREATING BACTERIAL AND VIRAL INFECTIONS WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1999-06-08 US disclosed
EP-0787720-A1 NOVEL PYRIDONECARBOXYLATE DERIVATIVE OR SALT THEREOF AND ANTIBACTERIAL CONTAINING THE SAME AS ACTIVE INGREDIENT WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1997-08-06 EP disclosed