SCHEMBL7009043

SCHEMBL7009043

FC(F)(F)c1ccc(-c2nc(Oc3ccnc(Cl)c3)cc(Oc3ccnc(Cl)c3)n2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 2/20 0.53
S1PR3 Q99500 1/20 0.53
TRPV1 Q8NER1 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
BLM P54132 2/20 0.39
FPR2 P25090 2/20 0.39
SCN9A Q15858 2/20 0.39
THRB P10828 1/20 0.38
HDAC4 P56524 1/20 0.38
ESR1 P03372 3/20 0.37
CASP3 P42574 2/20 0.37
KCNH2 Q12809 1/20 0.36
KDM4E B2RXH2 1/20 0.36
LMNA P02545 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
SENP8 Q96LD8 1/20 0.36
SENP7 Q9BQF6 1/20 0.36
SENP6 Q9GZR1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7006071 0.94 S1PR1 (0.48) S1PR1S1PR3TRPV1CYP1A2CYP2C9
SCHEMBL7009823 0.92 S1PR1 (0.48) S1PR1S1PR3TRPV1CYP1A2CYP2C9
SCHEMBL5252670 0.91 S1PR1 (0.52) S1PR1S1PR3TRPV1SCN9ATHRB
SCHEMBL7007490 0.89 S1PR1 (0.46) S1PR1S1PR3TRPV1FPR2SCN9A
SCHEMBL7004813 0.82 S1PR1 (0.43) S1PR1S1PR3TRPV1CYP1A2CYP2C9
SCHEMBL7008000 0.81 TRPV1 (0.49) S1PR1S1PR3TRPV1SCN9A
SCHEMBL7007712 0.81 S1PR1 (0.47) S1PR1S1PR3TRPV1CYP1A2CYP2C9
SCHEMBL30864860 0.80 KCNH2 (0.46) S1PR1S1PR3SCN9ATHRBKCNH2
SCHEMBL27314076 0.80 KCNH2 (0.46) S1PR1S1PR3SCN9ATHRBKCNH2
SCHEMBL8553275 0.79 GRM5 (0.41) S1PR1S1PR3TRPV1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0723960-B1 Herbicidal 2,6-disubstituted pyridines and 2,4-disubstituted pyrimidines BASF AG (DE) 2003-04-02 EP disclosed
US-5849758-A Herbicidal 2, 6-disubstituted pyridines and 2, 4-disubstituted pyrimidines AMERICAN CYANAMID COMPANY (US) 1998-12-15 US disclosed
EP-0823431-A1 Herbicidal 2,6-disubstituted pyridines and 2,4-disubstituted pyrimidines American Cyanamid Company (US) 1998-02-11 EP disclosed
EP-0723960-A1 Herbicidal 2,6-disubstituted pyridines and 2,4-disubstituted pyrimidines American Cyanamid Company (US) 1996-07-31 EP disclosed