SCHEMBL8553275

SCHEMBL8553275

N#Cc1cc(Oc2ccnc(Cl)c2)nc(-c2ccc(C(F)(F)F)cc2)c1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 2/20 0.41
S1PR1 P21453 1/20 0.41
S1PR3 Q99500 1/20 0.41
TRPV1 Q8NER1 1/20 0.41
KIF11 P52732 1/20 0.39
CTSS P25774 1/20 0.38
CTSK P43235 1/20 0.38
TOP1 P11387 2/20 0.36
PSD A5PKW4 1/20 0.35
BRAF P15056 1/20 0.34
KDR P35968 1/20 0.34
LTB4R Q15722 2/20 0.33
KCNH2 Q12809 2/20 0.33
DGAT1 O75907 1/20 0.33
SOAT1 P35610 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8549067 0.89 CTSS (0.45) GRM5CTSSCTSKKCNH2
SCHEMBL8553832 0.88 TRPV1 (0.43) TRPV1KIF11CTSSCTSKTOP1
SCHEMBL8552904 0.85 TRPV1 (0.39) TRPV1KIF11CTSSCTSKTOP1
SCHEMBL7004813 0.83 S1PR1 (0.43) S1PR1S1PR3TRPV1TOP1
SCHEMBL8552758 0.82 KIF11 (0.42) TRPV1KIF11CTSSCTSKKCNH2
SCHEMBL8548872 0.82 POLB (0.43) TRPV1KIF11CTSSCTSK
SCHEMBL7008000 0.81 TRPV1 (0.49) S1PR1S1PR3TRPV1
SCHEMBL8549675 0.80 ADORA1 (0.46) TRPV1KIF11CTSSCTSKKCNH2
SCHEMBL8471818 0.79 PSD (0.41) CTSSPSD
SCHEMBL7009043 0.79 S1PR1 (0.53) S1PR1S1PR3TRPV1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0820996-A1 Herbicidal cyanopyridines American Cyanamid Company (US) 1998-01-28 EP claimed
EP-0820996-A1 Herbicidal cyanopyridines American Cyanamid Company (US) 1998-01-28 EP disclosed