SCHEMBL7009792

SCHEMBL7009792

COc1ccc(N2CCN(CCn3cnc4sc(C(=O)N(C)C)c(C)c4c3=O)CC2)c(OC)c1

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 10/20 0.56
ADRA1D P25100 9/20 0.56
HTR1B P28222 9/20 0.56
ADRA1A P35348 9/20 0.56
ADRA1B P35368 9/20 0.56
CYP3A4 P08684 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
P2RX3 P56373 4/20 0.48
HTR7 P34969 1/20 0.47
KDM4E B2RXH2 1/20 0.45
TP53 P04637 1/20 0.44
MAPT P10636 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7012872 0.90 HTR1A (0.62) HTR1AADRA1DHTR1BADRA1AADRA1B
SCHEMBL7016146 0.83 HTR1A (0.51) HTR1AADRA1DHTR1BADRA1AADRA1B
SCHEMBL7012057 0.83 HTR1A (0.61) HTR1AADRA1DHTR1BADRA1AADRA1B
SCHEMBL7014998 0.83 HTR1A (0.61) HTR1AADRA1DHTR1BADRA1AADRA1B
SCHEMBL7007932 0.82 HTR1A (0.60) HTR1AADRA1DHTR1BADRA1AADRA1B
SCHEMBL7014563 0.82 HTR1A (0.53) HTR1AADRA1DHTR1BADRA1AADRA1B
SCHEMBL7014582 0.81 HTR1A (0.65) HTR1AADRA1DHTR1BADRA1AADRA1B
Water SCHEMBL7720208 0.81 HTR1A (0.64) HTR1AADRA1DHTR1BADRA1AADRA1B
SCHEMBL7015282 0.81 HTR1A (0.54) HTR1AADRA1DHTR1BADRA1AADRA1B
SCHEMBL7014231 0.80 HTR1A (0.63) HTR1AADRA1DHTR1BADRA1AADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0988306-B1 3-SUBSTITUTED 3,4 DIHYDRO-THIENO 2, 3-D]PYRIMIDINE DERIVATIVES AND PRODUCTION AND USE OF THE SAME ABBOTT GMBH & CO KG (DE) 2003-07-09 EP disclosed
US-6387912-B1 STROKE THERAPY BASF AKTIENGESELLSCHAFT (DE) 2002-05-14 US disclosed
US-6159962-A 3-substituted 3,4-dihydro-thieno[2,3-D]pyrimidine derivatives and production and use of the same BASF AKTIENGESELLSCHAFT (DE) 2000-12-12 US disclosed