SCHEMBL7010051

SCHEMBL7010051

CN1CCN(C(=O)c2ccc(B(O)O)cc2)CC1.O=C(O)c1ccc(B(O)O)cc1

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
POLB P06746 3/20 0.59
HPGD P15428 4/20 0.55
ALOX15 P16050 1/20 0.55
GRM5 P41594 1/20 0.55
KMT2A Q03164 3/20 0.52
MEN1 O00255 2/20 0.52
CYP1A2 P05177 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C19 P33261 1/20 0.52
NPC1 O15118 1/20 0.51
MKNK1 Q9BUB5 1/20 0.49
MKNK2 Q9HBH9 1/20 0.49
HRH3 Q9Y5N1 2/20 0.49
LMNA P02545 1/20 0.49
TSHR P16473 1/20 0.49
CYP2C9 P11712 1/20 0.48
EPHX2 P34913 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL532147 0.94 POLB (0.65) POLBHPGDALOX15GRM5KMT2A
Hydrochloric Acid SCHEMBL2550272 0.92 POLB (0.63) POLBHPGDALOX15GRM5KMT2A
SCHEMBL14980308 0.89 POLB (0.72) POLBHPGDALOX15GRM5KMT2A
SCHEMBL29253633 0.87 HPGD (0.61) POLBHPGDALOX15GRM5KMT2A
SCHEMBL7010056 0.86 L3MBTL1 (0.60) POLBHPGDALOX15GRM5KMT2A
SCHEMBL29950978 0.85 HPGD (0.57) POLBHPGDALOX15KMT2AMEN1
SCHEMBL10724841 0.82 POLB (0.81) POLBHPGDALOX15GRM5KMT2A
SCHEMBL9133746 0.80 ALDH1A1 (0.64) POLBHPGDKMT2AMEN1LMNA
SCHEMBL204078 0.79 HPGD (0.70) HPGDKMT2AMEN1LMNATSHR
SCHEMBL950365 0.79 HPGD (0.64) POLBHPGDKMT2AMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1296981-A2 SUBSTITUTED PYRROLOPYRIDINONE DERIVATIVES USEFUL AS PHOSPHODIESTERASE INHIBITORS Ortho-McNeil Pharmaceutical, Inc. (US) 2003-04-02 EP disclosed
WO-2001087882-A2 SUBSTITUTED PYRROLOPYRIDINONE DERIVATIVES USEFUL AS PHOSPHODIESTERASE INHIBITORS ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2001-11-22 WO disclosed