SCHEMBL7010219

SCHEMBL7010219

N#Cc1cc2ccccc2nc1-c1ccc(CBr)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.50
KDM4E B2RXH2 3/20 0.50
GAA P10253 2/20 0.50
LMNA P02545 1/20 0.49
THRB P10828 1/20 0.49
RXFP1 Q9HBX9 3/20 0.46
HTT P42858 1/20 0.46
HPGD P15428 3/20 0.43
PIP4K2A P48426 1/20 0.43
TSHR P16473 2/20 0.42
MAPT P10636 3/20 0.41
TP53 P04637 1/20 0.41
ALOX15 P16050 1/20 0.41
HBB P68871 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
PDE4B Q07343 1/20 0.41
PDE10A Q9Y233 1/20 0.41
KMT2A Q03164 2/20 0.39
MEN1 O00255 1/20 0.39
ADORA2A P29274 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3970132 0.76 ALDH1A1 (0.57) ALDH1A1KDM4EGAALMNATHRB
SCHEMBL14119232 0.74 KDM4E (0.58) ALDH1A1KDM4EGAALMNATHRB
SCHEMBL30804565 0.72 TSHR (0.55) ALDH1A1KDM4EGAALMNATHRB
SCHEMBL30804559 0.72 TSHR (0.55) ALDH1A1KDM4EGAALMNATHRB
SCHEMBL1939347 0.71 NPSR1 (0.56) ALDH1A1KDM4ELMNATHRBRXFP1
SCHEMBL13762566 0.71 CNR1 (0.49) ALDH1A1KDM4ELMNATHRBRXFP1
SCHEMBL7683450 0.71 CNR2 (0.47) ALDH1A1KDM4EGAAHPGDSMN1; SMN2
SCHEMBL7014505 0.71 ALDH1A1 (0.62) ALDH1A1KDM4EGAALMNATHRB
SCHEMBL30804562 0.70 KDM4E (0.53) ALDH1A1KDM4EGAALMNATHRB
SCHEMBL4436697 0.70 ALDH1A1 (0.61) ALDH1A1KDM4EGAALMNATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1327631-A2 Fused heterocyclic compounds, their production and use as angiotensin II antagonists Takeda Chemical Industries, Ltd. (JP) 2003-07-16 EP disclosed
EP-0518033-B1 Fused heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-07-02 EP disclosed
US-5389641-A Fused heterocyclic compounds, having angiotensin II antagonistic activity TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-02-14 US disclosed
EP-0518033-A1 Fused heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-12-16 EP disclosed