SCHEMBL7010433

SCHEMBL7010433

O=C(c1ccc(CBr)cc1)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.65

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 3/20 0.65
GSK3B P49841 2/20 0.59
PTPN1 P18031 2/20 0.59
CES2 O00748 2/20 0.53
CES1 P23141 2/20 0.53
VNN1 O95497 3/20 0.50
EPHX2 P34913 1/20 0.49
MAOB P27338 2/20 0.46
LSS P48449 1/20 0.44
CYP2C8 P10632 1/20 0.44
MMP1 P03956 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27932511 0.85 SRD5A2 (0.86) SRD5A2GSK3BPTPN1CES2CES1
SCHEMBL187134 0.84 CES2 (0.61) SRD5A2CES2CES1
SCHEMBL4229 0.84 TAAR1 (0.54) SRD5A2GSK3BPTPN1MAOB
SCHEMBL9541276 0.84 CES2 (0.61) SRD5A2CES2CES1
SCHEMBL648641 0.84 SRD5A2 (0.83) SRD5A2GSK3BPTPN1CES2CES1
Ammonia Solution, Strong SCHEMBL28278225 0.82 TAAR1 (0.52) SRD5A2GSK3BPTPN1MAOB
Hydrochloric Acid SCHEMBL27733522 0.82 SRD5A2 (0.79) SRD5A2GSK3BPTPN1CES2CES1
SCHEMBL2685467 0.79 SRD5A2 (0.68) SRD5A2GSK3BPTPN1CES2CES1
SCHEMBL2976204 0.79 PTPN1 (0.55) PTPN1CES2CES1VNN1
SCHEMBL13410662 0.78 SRD5A2 (0.73) SRD5A2GSK3BPTPN1CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
US-5753664-A ANTITUMOR AGENTS, PYRIMIDONES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-05-19 US disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed