SCHEMBL7011905

SCHEMBL7011905

COc1ccc([N+](=O)[O-])cc1OCCN1CCN(C(=O)OC(C)(C)C)CC1

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.53
LMNA P02545 2/20 0.53
MAPT P10636 1/20 0.53
SMN1; SMN2 Q16637 2/20 0.48
HRH2 P25021 1/20 0.46
HRH1 P35367 1/20 0.46
DRD3 P35462 2/20 0.45
KDM4E B2RXH2 1/20 0.45
KMT2A Q03164 3/20 0.44
DRD2 P14416 1/20 0.44
MEN1 O00255 1/20 0.44
HPGD P15428 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43
SLC9A1 P19634 1/20 0.43
HTR1A P08908 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12448368 0.95 ALDH1A1 (0.52) ALDH1A1LMNAMAPTSMN1; SMN2HRH2
SCHEMBL22117865 0.88 ALDH1A1 (0.53) ALDH1A1LMNAMAPTSMN1; SMN2HRH2
SCHEMBL22118025 0.86 ALDH1A1 (0.51) ALDH1A1LMNAMAPTSMN1; SMN2HRH2
SCHEMBL7005111 0.83 DRD3 (0.48) ALDH1A1DRD3DRD2RXFP1
SCHEMBL18910916 0.83 MAPT (0.52) ALDH1A1LMNAMAPTSMN1; SMN2HRH2
SCHEMBL16570456 0.83 HRH2 (0.64) ALDH1A1LMNAMAPTHRH2HRH1
SCHEMBL21644472 0.82 ALDH1A1 (0.50) ALDH1A1LMNAMAPT
SCHEMBL25398475 0.82 ALDH1A1 (0.55) ALDH1A1LMNAMAPTSMN1; SMN2HRH2
SCHEMBL1929880 0.81 LTA4H (0.57) ALDH1A1LMNAMAPTSMN1; SMN2KDM4E
SCHEMBL15244045 0.81 ALDH1A1 (0.49) ALDH1A1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1309551-A1 INDOLINE DERIVATIVES AS 5HT2C ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 2003-05-14 EP disclosed
WO-2002014273-A1 INDOLINE DERIVATIVES AS 5HT2C ANTAGONISTS SMITHKLINE BEECHAM P.L.C. (GB) 2002-02-21 WO disclosed