Bicarbonate

Bicarbonate

SCHEMBL7013221

O=C(O)O.O=[N+]([O-])c1cc2c(NCc3ccccc3)nc(C3CCCCC3)nc2s1

nearest known ligand 0.55

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3A known ✓ P49840 1/20 0.37
GSK3B known ✓ P49841 1/20 0.37
PDE5A O76074 5/20 0.55
PDE10A Q9Y233 1/20 0.41
CHRM3 P20309 1/20 0.40
PDE4A P27815 1/20 0.40
PDE4B Q07343 1/20 0.40
PDE4C Q08493 1/20 0.40
PDE4D Q08499 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
MAPT P10636 2/20 0.39
ALDH1A1 P00352 1/20 0.39
POLB P06746 1/20 0.39
F2 P00734 1/20 0.38
THRB P10828 1/20 0.38
CDK2 P24941 2/20 0.37
USP1 O94782 1/20 0.37
WDR48 Q8TAF3 1/20 0.37
DYRK1A Q13627 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7427837 0.97 PDE5A (0.58) PDE5APDE10ACHRM3PDE4APDE4B
Bicarbonate SCHEMBL7014883 0.92 PDE5A (0.46) PDE5APDE4APDE4BPDE4CPDE4D
Bicarbonate SCHEMBL7021236 0.92 PDE5A (0.45) PDE5AALDH1A1POLBUSP1WDR48
Bicarbonate SCHEMBL7018347 0.91 PDE5A (0.44) PDE5AMEN1KMT2AMAPTCDK2
SCHEMBL8179646 0.90 PDE5A (0.44) PDE5APDE10ACHRM3PDE4APDE4B
Bicarbonate SCHEMBL7020472 0.88 PDE5A (0.42) PDE5APDE10APDE4APDE4BPDE4C
Bicarbonate SCHEMBL7018662 0.87 ALDH1A1 (0.47) PDE5APDE4APDE4BPDE4CPDE4D
Bicarbonate SCHEMBL7013300 0.86 ACHE (0.42) PDE5AMEN1KMT2AMAPTALDH1A1
Bicarbonate SCHEMBL7017039 0.84 PDE5A (0.59) PDE5APDE10ACHRM3PDE4APDE4B
Bicarbonate SCHEMBL7011719 0.84 PDE5A (0.59) PDE5APDE10ACHRM3PDE4APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0934321-B1 THIENOPYRIMIDINE WITH PHOSPHODIESTERASE V INHIBITING EFFECT MERCK PATENT GMBH (DE) 2003-08-06 EP disclosed