SCHEMBL7014154

SCHEMBL7014154

c1csc(C2CCCNC2)c1

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 1/20 0.45
DRD2 P14416 1/20 0.45
DRD3 P35462 1/20 0.45
CHEK1 O14757 1/20 0.43
CCNA2 P20248 1/20 0.43
CDK2 P24941 1/20 0.43
CCNA1 P78396 1/20 0.43
KCNH2 Q12809 2/20 0.41
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
CYP2D6 P10635 1/20 0.40
SLC6A2 P23975 1/20 0.40
SLC6A4 P31645 1/20 0.40
SLC6A3 Q01959 1/20 0.40
POLB P06746 1/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3648603 0.89 HTR3A (0.44) POLBGAAMAPT
SCHEMBL8133890 0.82
SCHEMBL498606 0.82 MAPT (0.47) CYP2D6POLBGAAMAPT
SCHEMBL5467244 0.80 SLC18A3 (0.48) HTR2CPOLBGAAMAPT
SCHEMBL663162 0.80 MAPT (0.46) CYP2D6POLBGAAMAPT
SCHEMBL930295 0.80 MAPT (0.46) CYP2D6POLBGAAMAPT
Hydrochloric Acid SCHEMBL2803164 0.79 SLC18A3 (0.47) HTR2CPOLBGAAMAPT
SCHEMBL7122480 0.78 MAPT (0.44) CYP2D6POLBGAAMAPT
SCHEMBL497608 0.77
Hydrochloric Acid SCHEMBL11286601 0.75

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104703970-A Substituted carbamate compounds and their use as transient receptor potential (TRP) channel antagonists HOFFMANN LA ROCHE 2015-06-10 CN disclosed
CN-1419545-A 3-cyanoquinolines, 3-cyano-1,6-naphthyridines, and 3-cyano-1,7-naphthyridines as protein kinase inhibitors WYETH CORP (US) 2003-05-21 CN disclosed
EP-1268431-A1 3-CYANOQUINOLINES,3-CYANO-1,6-NAPHTHYRIDINES, AND 3-CYANO-1,7-NAPHTHYRIDINES AS PROTEIN KINASE INHIBITORS Wyeth (US) 2003-01-02 EP disclosed
WO-2001072711-A1 3-CYANOQUINOLINES,3-CYANO-1,6-NAPHTHYRIDINES, AND 3-CYANO-1,7-NAPHTHYRIDINES AS PROTEIN KINASE INHIBITORS WYETH (US) 2001-10-04 WO disclosed