SCHEMBL7014394

SCHEMBL7014394

Brc1ccc2c(Nc3ccc(Oc4ccccc4)cc3)ccnc2c1

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 8/20 0.78
ERBB2 P04626 1/20 0.71
GAK O14976 3/20 0.56
EGFR P00533 4/20 0.53
HTT P42858 1/20 0.52
FGFR2 P21802 1/20 0.47
RIPK2 O43353 3/20 0.46
EPHB2 P29323 1/20 0.46
GAA P10253 2/20 0.46
MAPT P10636 2/20 0.46
POLB P06746 1/20 0.46
NTSR1 P30989 1/20 0.46
RAD52 P43351 1/20 0.46
RECQL P46063 1/20 0.46
BLM P54132 1/20 0.46
KMT2A Q03164 1/20 0.46
PAX8 Q06710 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3321525 0.85 ERBB2 (0.71) ALKERBB2GAKEGFRHTT
SCHEMBL1387165 0.84 ERBB2 (1.00) ALKERBB2GAKEGFRHTT
Hydrochloric Acid SCHEMBL8812168 0.82 ERBB2 (0.97) ALKERBB2GAKEGFRHTT
SCHEMBL7015701 0.82 ALK (0.78) ALKERBB2GAKEGFRRIPK2
SCHEMBL10000194 0.81 ERBB2 (0.94) ALKERBB2GAKEGFRHTT
SCHEMBL8809979 0.79 FGFR2 (0.72) ERBB2GAKEGFRHTTFGFR2
SCHEMBL19633677 0.79 ALK (0.67) ALKERBB2GAKEGFRHTT
SCHEMBL19633717 0.78 ALK (0.81) ALKGAKEGFR
Hydrochloric Acid SCHEMBL8933873 0.78 FGFR2 (0.70) ERBB2GAKEGFRHTTFGFR2
SCHEMBL28133700 0.77 ERBB2 (0.71) ALKERBB2GAKEGFRHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1268431-A1 3-CYANOQUINOLINES,3-CYANO-1,6-NAPHTHYRIDINES, AND 3-CYANO-1,7-NAPHTHYRIDINES AS PROTEIN KINASE INHIBITORS Wyeth (US) 2003-01-02 EP disclosed
WO-2001072711-A1 3-CYANOQUINOLINES,3-CYANO-1,6-NAPHTHYRIDINES, AND 3-CYANO-1,7-NAPHTHYRIDINES AS PROTEIN KINASE INHIBITORS WYETH (US) 2001-10-04 WO disclosed