SCHEMBL7014783

SCHEMBL7014783

O=c1[nH]c2occc2c(=O)n1CCC(S)CS

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.33
ALDH1A1 P00352 4/20 0.33
HPGD P15428 2/20 0.33
KDM4E B2RXH2 2/20 0.32
MAPK1 P28482 1/20 0.31
HSD17B10 Q99714 1/20 0.31
MEN1 O00255 1/20 0.30
POLB P06746 1/20 0.30
PKM P14618 1/20 0.30
KMT2A Q03164 1/20 0.30
MPO P05164 1/20 0.30
CYP1A2 P05177 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7014787 1.00 TSHR (0.33) TSHRALDH1A1HPGDKDM4EMAPK1
SCHEMBL7019442 0.86 TSHR (0.35) TSHRALDH1A1HPGDKDM4EMEN1
SCHEMBL7019436 0.86 TSHR (0.35) TSHRALDH1A1HPGDKDM4EMEN1
SCHEMBL7014980 0.74 TSHR (0.32) TSHRALDH1A1HPGDKDM4EMPO
SCHEMBL7014984 0.74 TSHR (0.32) TSHRALDH1A1HPGDKDM4EMPO
SCHEMBL7019417 0.73 FEN1 (0.50) ALDH1A1KDM4EHSD17B10POLBPKM
SCHEMBL7019413 0.73 FEN1 (0.50) ALDH1A1KDM4EHSD17B10POLBPKM
SCHEMBL7022632 0.72 XDH (0.41) ALDH1A1HPGDKDM4EHSD17B10
SCHEMBL7023095 0.72 ADORA3 (0.32) ALDH1A1HPGDKDM4EHSD17B10
SCHEMBL7022638 0.72 XDH (0.41) ALDH1A1HPGDKDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1357114-A1 Substituted pyrimidin-2,4(1H,3H)-diones as inhibitors of Matrix Metalloproteinases (MMP) IBFB GmbH Privates Institut für biomedizinische Forschung und Beratung (DE) 2003-10-29 EP disclosed