SCHEMBL7015014

SCHEMBL7015014

O=Cc1ccc(C(=O)c2ccc(Cl)nc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAPRT Q6XQN6 1/20 0.55
ALDH1A1 P00352 3/20 0.46
DGAT1 O75907 1/20 0.43
SMN1; SMN2 Q16637 3/20 0.42
GAA P10253 2/20 0.42
RAB9A P51151 2/20 0.42
L3MBTL1 Q9Y468 1/20 0.41
HSD17B10 Q99714 1/20 0.41
KCNQ3 O43525 2/20 0.41
KCNQ2 O43526 2/20 0.41
KCNE1 P15382 2/20 0.41
KCNQ1 P51787 2/20 0.41
MEN1 O00255 1/20 0.40
LMNA P02545 1/20 0.40
KMT2A Q03164 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
MDM4 O15151 1/20 0.40
TP53 P04637 1/20 0.40
MDM2 Q00987 1/20 0.40
EGFR P00533 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7440808 0.85 NAPRT (0.72) NAPRTDGAT1SMN1; SMN2GAARAB9A
SCHEMBL2475597 0.82 NAPRT (0.62) NAPRTDGAT1SMN1; SMN2GAARAB9A
SCHEMBL3383611 0.80 NAPRT (0.66) NAPRTALDH1A1DGAT1SMN1; SMN2GAA
SCHEMBL31473447 0.80 NAPRT (0.66) NAPRTALDH1A1DGAT1SMN1; SMN2GAA
SCHEMBL6852409 0.79 ALDH1A1 (0.68) ALDH1A1HSD17B10LMNAEGFR
SCHEMBL4467915 0.79 NPC1 (0.62) NAPRTALDH1A1DGAT1SMN1; SMN2GAA
SCHEMBL17676098 0.79 RAB9A (0.64) NAPRTALDH1A1DGAT1SMN1; SMN2GAA
SCHEMBL5305773 0.79 NAPRT (0.58) NAPRTDGAT1SMN1; SMN2GAARAB9A
SCHEMBL29457431 0.79 NPC1 (0.62) NAPRTALDH1A1DGAT1SMN1; SMN2GAA
SCHEMBL3565290 0.77 HSD17B10 (0.70) ALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
US-5753664-A ANTITUMOR AGENTS, PYRIMIDONES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-05-19 US disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed