SCHEMBL7015547

SCHEMBL7015547

O=C(c1ccc(Cl)cc1)c1cccc(CBr)c1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 2/20 0.47
MAPK1 P28482 1/20 0.47
MRGPRX4 Q96LA9 1/20 0.47
MEP1A Q16819 1/20 0.46
MEP1B Q16820 1/20 0.46
GSK3B P49841 1/20 0.46
CNR2 P34972 1/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
ATM Q13315 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
MAPT P10636 1/20 0.45
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
CES2 O00748 2/20 0.43
CES1 P23141 2/20 0.43
HPGD P15428 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20836220 0.88 CES2 (0.56) SRD5A2MEP1BL3MBTL1ATMTDP1
SCHEMBL185962 0.88 ATM (0.52) SRD5A2MEP1AMEP1BCNR2L3MBTL1
SCHEMBL29572523 0.88 ATM (0.52) SRD5A2MEP1AMEP1BCNR2L3MBTL1
SCHEMBL435297 0.86 L3MBTL1 (0.63) SRD5A2CNR2L3MBTL1ATMTDP1
SCHEMBL29728644 0.86 L3MBTL1 (0.63) SRD5A2CNR2L3MBTL1ATMTDP1
SCHEMBL11493619 0.83 MEP1B (0.46) SRD5A2MAPK1MEP1BL3MBTL1ATM
SCHEMBL14302252 0.83 SRD5A2 (0.47) SRD5A2MAPK1MRGPRX4CNR2L3MBTL1
SCHEMBL2931832 0.83 CES2 (0.51) L3MBTL1ATMTDP1CES2CES1
SCHEMBL1744667 0.82 SRD5A2 (0.57) SRD5A2MAPK1GSK3BL3MBTL1MAPT
SCHEMBL11541766 0.82 L3MBTL1 (0.47) SRD5A2MAPK1MRGPRX4CNR2L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
US-5753664-A ANTITUMOR AGENTS, PYRIMIDONES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-05-19 US disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed
EP-0151529-B1 5-(AMINO OR SUBSTITUTED AMINO)-1,2,3-TRIAZOLES MERCK & CO. INC. (US) 1991-09-18 EP disclosed
US-4590201-A ANTICOCCIDIAL AGENT FOR ANIMALS PARTICULARLY FOR POULTRY MERCK & CO., INC. (US) 1986-05-20 US disclosed
EP-0151529-A2 5-(Amino or substituted amino)-1,2,3-triazoles MERCK & CO. INC. (US) 1985-08-14 EP disclosed
US-4192890-A Novel benzoylphenylacetic acid esters ROUSSEL UCLAF (FR) 1980-03-11 US disclosed
US-3995056-A Butyric acid derivatives for treating pain and inflammation ROUSSEL-UCLAF (FR) 1976-11-30 US disclosed
US-3931302-A ANTIINFLAMMATORY, ANALGESIC ROUSSEL-UCLAF (FR) 1976-01-06 US disclosed