SCHEMBL7016308

SCHEMBL7016308

CCn1c(SC)nc2c(ccn2Cc2ccc(C(=O)c3ccc(OCCN(C)C)cc3)cc2)c1=O

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.39
CDK4 P11802 1/20 0.38
CCND1 P24385 1/20 0.38
CCND2 P30279 1/20 0.38
CCND3 P30281 1/20 0.38
BCHE P06276 4/20 0.37
ACHE P22303 4/20 0.37
P2RX3 P56373 1/20 0.37
USP1 O94782 3/20 0.36
HRH3 Q9Y5N1 2/20 0.36
DRD2 P14416 1/20 0.36
DRD3 P35462 1/20 0.36
TP53 P04637 1/20 0.35
MAPT P10636 1/20 0.35
TSHR P16473 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7012711 0.84 PSMB1 (0.49) BCHEACHEHRH3MAPTTSHR
SCHEMBL7019933 0.83 HDAC1 (0.41) CYP19A1TP53MAPTTSHRRXFP1
SCHEMBL7017888 0.83 TP53 (0.47) P2RX3TP53MAPTTSHRRXFP1
Hydrochloric Acid SCHEMBL7016880 0.83 SMN1; SMN2 (0.46) BCHEACHEMAPT
SCHEMBL7010029 0.82 TP53 (0.36) CYP19A1P2RX3TP53MAPTTSHR
SCHEMBL7015187 0.80 RAB9A (0.37) CYP19A1P2RX3MAPTTSHRPOLB
SCHEMBL7015809 0.79 HDAC6 (0.48) TP53MAPTTSHR
Hydrochloric Acid SCHEMBL7012709 0.78 SRC (0.37) P2RX3TP53MAPTTSHRRXFP1
Hydrochloric Acid SCHEMBL7016878 0.77 SRC (0.39) P2RX3HRH3TP53MAPTTSHR
SCHEMBL7008875 0.74 TP53 (0.42) P2RX3TP53MAPTTSHRRXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed