SCHEMBL7016775

SCHEMBL7016775

CCn1c(S)nc2cccc(C)c2c1=O

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ELANE P08246 12/20 0.46
CASR P41180 2/20 0.45
PIK3CD O00329 1/20 0.44
PARP1 P09874 1/20 0.43
LMNA P02545 2/20 0.41
GAA P10253 1/20 0.41
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40
MAPK1 P28482 1/20 0.40
HSD17B10 Q99714 1/20 0.40
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11923470 0.82 PIK3CD (0.50) ELANECASRPIK3CDPARP1LMNA
SCHEMBL7011912 0.80 ELANE (0.46) ELANECASRPIK3CDPARP1
SCHEMBL9670265 0.76 KDM4E (0.60) LMNAGAAKDM4EALDH1A1HPGD
SCHEMBL9670318 0.75 PIK3CD (0.49) ELANECASRPIK3CDPARP1LMNA
SCHEMBL28451245 0.72 PIK3CD (0.50) ELANECASRPIK3CDPARP1LMNA
SCHEMBL20081332 0.71 NPC1 (0.62) CASRPIK3CDLMNAGAAKDM4E
SCHEMBL7014708 0.69 ELANE (0.49) ELANECASRPIK3CDPARP1LMNA
SCHEMBL1129587 0.69 PIK3CG (0.51) ELANEPIK3CDLMNAKDM4EALDH1A1
SCHEMBL16796581 0.69 TLR8 (0.55) CASRLMNAGAAKDM4EALDH1A1
SCHEMBL13804449 0.69 TRPA1 (0.51) ELANEPARP1ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
US-5753664-A ANTITUMOR AGENTS, PYRIMIDONES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-05-19 US disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed