SCHEMBL9670265

SCHEMBL9670265

CCn1c(S)nc2ccccc2c1=O

nearest known ligand 0.60

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.60
MAPK1 P28482 3/20 0.60
RAB9A P51151 2/20 0.55
LMNA P02545 4/20 0.53
GAA P10253 1/20 0.53
MEN1 O00255 7/20 0.52
KMT2A Q03164 7/20 0.52
MAPT P10636 4/20 0.52
ALDH1A1 P00352 2/20 0.52
GFER P55789 1/20 0.52
TSHR P16473 3/20 0.50
HPGD P15428 2/20 0.50
HSD17B10 Q99714 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
ATM Q13315 1/20 0.50
POLB P06746 2/20 0.49
NPC1 O15118 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24340312 0.87 ALDH1A1 (0.51) KDM4EMAPK1LMNAGAAMEN1
SCHEMBL10739963 0.84 ALDH1A1 (0.60) KDM4ELMNAGAAMEN1KMT2A
SCHEMBL9670541 0.83 ALDH1A1 (0.68) KDM4EMAPK1RAB9ALMNAGAA
SCHEMBL14010912 0.82 ALDH1A1 (0.66) KDM4ERAB9ALMNAGAAMEN1
SCHEMBL8347824 0.81 MEN1 (0.68) KDM4EMAPK1RAB9ALMNAGAA
SCHEMBL14363850 0.80 KDM4E (0.60) KDM4EMAPK1RAB9ALMNAGAA
SCHEMBL2994370 0.80 KDM4E (0.60) KDM4EMAPK1RAB9ALMNAGAA
SCHEMBL9671285 0.80 MEN1 (0.69) KDM4ERAB9ALMNAGAAMEN1
SCHEMBL9724531 0.80 TDP1 (0.59) KDM4EMAPK1LMNAGAAMEN1
SCHEMBL31621465 0.80 TDP1 (0.59) KDM4EMAPK1LMNAGAAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0276825-B1 4 (3H)-QUINAZOLINONE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS NISSHIN FLOUR MILLING CO., LTD. (JP) 1992-09-09 EP disclosed
EP-0276826-B1 2-ALKYLSULFINYL-4 (3H)-QUINAZOLINONE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS NISSHIN FLOUR MILLING CO., LTD. (JP) 1991-12-27 EP disclosed
US-5008266-A Antiulcer agent NISSHIN FLOUR MILLING CO., LTD. (JP) 1991-04-16 US disclosed
US-4861780-A 4(3H)-quinazolinone derivatives and pharmaceutical compositions NISSHIN FLOUR MILLING CO., LTD. (JP) 1989-08-29 US disclosed
US-4833144-A ANTIULCER AGENTS NISSHIN FLOUR MILLING CO., LTD. (JP) 1989-05-23 US disclosed
EP-0276826-A1 2-Alkylsulfinyl-4 (3H)-quinazolinone derivatives, processes for their preparation and pharmaceutical compositions NISSHIN FLOUR MILLING CO., LTD. (JP) 1988-08-03 EP disclosed
EP-0276825-A1 4 (3H)-Quinazolinone derivatives, processes for their preparation and pharmaceutical compositions NISSHIN FLOUR MILLING CO., LTD. (JP) 1988-08-03 EP disclosed