SCHEMBL7016776

SCHEMBL7016776

C=CCOC(=O)Nc1cccc(C(CC)N(C(=O)OC(C)(C)C)c2cc(N3CCOCC3)cc(COC3CCCCO3)n2)c1

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CASR P41180 7/20 0.35
NPY1R P25929 2/20 0.33
KCNH2 Q12809 1/20 0.33
SPHK1 Q9NYA1 1/20 0.32
EGFR P00533 4/20 0.31
NPC1 O15118 1/20 0.30
MAPT P10636 1/20 0.30
RAB9A P51151 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
AKT1 P31749 1/20 0.30
KIF18A Q8NI77 1/20 0.30
RXFP1 Q9HBX9 1/20 0.30
FKBP1A P62942 1/20 0.30
BTK Q06187 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7011740 0.93 CASR (0.36) CASRNPY1RKCNH2SPHK1EGFR
SCHEMBL7016255 0.83 ALDH1A1 (0.34) MAPTSMN1; SMN2
SCHEMBL7017114 0.81 CASR (0.37) CASRNPY1RKCNH2SPHK1EGFR
SCHEMBL7017580 0.79 NPY1R (0.37) NPY1RKCNH2
SCHEMBL7012036 0.77 ZAP70 (0.32)
SCHEMBL7016596 0.77 NPY1R (0.34) CASRNPY1RKCNH2
SCHEMBL7012030 0.77 NPY1R (0.34) CASRNPY1RKCNH2
SCHEMBL7011470 0.77 NPY1R (0.35) CASRNPY1RKCNH2SPHK1
SCHEMBL7011382 0.73 JAK3 (0.39) NPC1MAPTRAB9ASMN1; SMN2AKT1
SCHEMBL7011391 0.73 JAK2 (0.36) NPY1RKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0889034-B1 AMINOPYRIDINE DERIVATIVES BANYU PHARMA CO LTD (JP) 2003-09-17 EP disclosed
US-6011039-A USEFUL AS NEUROPEPTIDE Y RECEPTOR ANTAGONISTS; TREATING HYPERPHAGIA, OBESITY OR DIABETES BANYU PHARMACEUTICAL CO., LTD. (JP) 2000-01-04 US disclosed
EP-0889034-A1 AMINOPYRIDINE DERIVATIVES BANYU PHARMACEUTICAL CO., LTD. (JP) 1999-01-07 EP disclosed