SCHEMBL7016909

SCHEMBL7016909

CC(C)[Si](C(C)C)(C(C)C)n1cc(C2CCN(C)CC2)c2cc(-c3ccc(Cl)cc3)ccc21

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 14/20 0.53
HTR6 P50406 2/20 0.45
HTR1B P28222 1/20 0.45
DRD4 P21917 1/20 0.42
HTR2A P28223 1/20 0.41
SLC6A4 P31645 1/20 0.36
MAPK11 Q15759 1/20 0.36
MAPK14 Q16539 1/20 0.36
IKBKB O14920 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7710645 0.90 DRD2 (0.54) DRD2HTR6HTR1BHTR2A
SCHEMBL7018674 0.87 DRD2 (0.51) DRD2HTR6HTR1BHTR2A
SCHEMBL6642794 0.81 DRD2 (0.43) DRD2HTR6HTR1BHTR2ASLC6A4
SCHEMBL8182800 0.79 DRD2 (0.41) DRD2HTR6HTR1BHTR2ASLC6A4
SCHEMBL7019936 0.78 HTR6 (0.41) DRD2HTR6HTR2ASLC6A4
SCHEMBL7016982 0.78 CHRM2 (0.43) DRD2HTR6HTR1BHTR2ASLC6A4
SCHEMBL12128118 0.77 APP (0.46) DRD2HTR6HTR1B
SCHEMBL27516823 0.76 DRD2 (0.50) DRD2HTR6HTR1BDRD4HTR2A
SCHEMBL12127438 0.74 DRD2 (0.39) DRD2HTR6HTR1BSLC6A4
SCHEMBL12127481 0.74 HTR1B (0.46) DRD2HTR6HTR1BSLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1089993-B1 5-HT1F AGONISTS LILLY CO ELI (US) 2003-10-22 EP disclosed
EP-1089993-A1 5-HT1F AGONISTS ELI LILLY AND COMPANY (US) 2001-04-11 EP disclosed
WO-2000000487-A1 5-HT1F AGONISTS ELI LILLY AND COMPANY (US) 2000-01-06 WO disclosed