SCHEMBL7017707

SCHEMBL7017707

NCc1cccc(C2C[C@@H]2C(N)=O)c1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SLC9A1 P19634 4/20 0.46
ALDH1A1 P00352 3/20 0.41
NOS3 P29474 2/20 0.41
NOS1 P29475 2/20 0.41
NOS2 P35228 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
ENPP2 Q13822 1/20 0.41
CYP3A4 P08684 1/20 0.41
NFKB1 P19838 1/20 0.41
KDM1A O60341 3/20 0.40
LOXL2 Q9Y4K0 2/20 0.40
MAOA P21397 2/20 0.40
CYP4F2 P78329 2/20 0.40
CYP4A11 Q02928 2/20 0.40
MAOB P27338 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7019552 0.84 PRMT6 (0.39) ALDH1A1NOS3NOS1NOS2SMN1; SMN2
SCHEMBL7019556 0.84 PRMT6 (0.39) ALDH1A1NOS3NOS1NOS2SMN1; SMN2
SCHEMBL15540612 0.78 SLC9A1 (0.71) SLC9A1ALDH1A1
SCHEMBL4134867 0.78 KDM1A (0.59) SLC9A1ALDH1A1KDM1A
SCHEMBL4133997 0.78 HTR2A (0.51) SLC9A1ALDH1A1
SCHEMBL24737580 0.78 SLC9A1 (0.71) SLC9A1ALDH1A1
SCHEMBL4133995 0.78 HTR2A (0.51) SLC9A1ALDH1A1
SCHEMBL24737578 0.78 SLC9A1 (0.71) SLC9A1ALDH1A1
SCHEMBL24737867 0.78 SLC9A1 (0.71) SLC9A1ALDH1A1
SCHEMBL4134864 0.78 KDM1A (0.59) SLC9A1ALDH1A1KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1368341-A1 PHENYL DERIVATIVES 3 MERCK PATENT GmbH (DE) 2003-12-10 EP disclosed
WO-2002074765-A1 PHENYL DERIVATIVES 3 MERCK PATENT GMBH (DE) 2002-09-26 WO disclosed