SCHEMBL7019556

SCHEMBL7019556

NCc1cccc(C2CCC[C@@H]2C(N)=O)c1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PRMT6 Q96LA8 1/20 0.39
HRH3 Q9Y5N1 2/20 0.38
ALDH1A1 P00352 2/20 0.38
NOS3 P29474 2/20 0.38
NOS1 P29475 2/20 0.38
NOS2 P35228 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
CYP3A4 P08684 1/20 0.38
NFKB1 P19838 1/20 0.38
SIRT2 Q8IXJ6 1/20 0.38
SIRT1 Q96EB6 1/20 0.38
TPSAB1 Q15661 1/20 0.38
ENPP2 Q13822 1/20 0.38
LOXL2 Q9Y4K0 2/20 0.37
CFD P00746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7019552 1.00 PRMT6 (0.39) PRMT6HRH3ALDH1A1NOS3NOS1
SCHEMBL7017707 0.84 SLC9A1 (0.46) ALDH1A1NOS3NOS1NOS2SMN1; SMN2
SCHEMBL4607572 0.79 GRIA4 (0.47) SIRT2SIRT1
SCHEMBL4606839 0.78 KCNQ3 (0.50) HRH3ALDH1A1SIRT2SIRT1
SCHEMBL3323648 0.75 KCNQ3 (0.54) HRH3ALDH1A1
SCHEMBL25359641 0.73 PRMT6 (0.44) PRMT6TPSAB1ENPP2LOXL2
SCHEMBL30531117 0.73 PRMT6 (0.44) PRMT6TPSAB1ENPP2LOXL2
SCHEMBL4608450 0.72 GRIA4 (0.46) SMN1; SMN2SIRT2SIRT1
Formic Acid SCHEMBL27536013 0.72 TPSAB1 (0.45) CYP3A4TPSAB1ENPP2
Hydrochloric Acid SCHEMBL15922780 0.72 TPSAB1 (0.43) PRMT6TPSAB1ENPP2LOXL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1368341-A1 PHENYL DERIVATIVES 3 MERCK PATENT GmbH (DE) 2003-12-10 EP claimed
WO-2002074765-A1 PHENYL DERIVATIVES 3 MERCK PATENT GMBH (DE) 2002-09-26 WO claimed
EP-1368341-A1 PHENYL DERIVATIVES 3 MERCK PATENT GmbH (DE) 2003-12-10 EP disclosed
WO-2002074765-A1 PHENYL DERIVATIVES 3 MERCK PATENT GMBH (DE) 2002-09-26 WO disclosed