Triaziquone

Triaziquone

SCHEMBL7017795

C[SiH](C)O[SiH3].O=C1C=C(N2CC2)C(=O)C(N2CC2)=C1N1CC1

nearest known ligand 0.39

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.39
HTT P42858 2/20 0.39
TP53 P04637 1/20 0.39
STAT3 P40763 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
DNMT1 P26358 1/20 0.38
APAF1 O14727 2/20 0.32
TDP2 O95551 2/20 0.32
NSD2 O96028 2/20 0.32
HKDC1 Q2TB90 2/20 0.32
KMT2A Q03164 2/20 0.30
MEN1 O00255 1/20 0.30
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30
GALK1 P51570 1/20 0.30
BLM P54132 1/20 0.30
ATM Q13315 1/20 0.30
NOD2 Q9HC29 1/20 0.30
ATG4B Q9Y4P1 1/20 0.30
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Triaziquone SCHEMBL21835057 0.88 MAPT (0.44) MAPTHTTTP53STAT3SMN1; SMN2
Triaziquone SCHEMBL21811697 0.84 MAPT (0.42) MAPTHTTTP53STAT3SMN1; SMN2
Triaziquone SCHEMBL8303 0.84 DNMT1 (0.48) MAPTHTTTP53STAT3SMN1; SMN2
Triaziquone SCHEMBL11039269 0.82 MAPT (0.43) MAPTHTTTP53STAT3SMN1; SMN2
Triaziquone SCHEMBL149876 0.82 MAPT (0.46) MAPTHTTTP53STAT3SMN1; SMN2
Triaziquone SCHEMBL7783197 0.82 MAPT (0.46) MAPTHTTTP53STAT3SMN1; SMN2
Triaziquone SCHEMBL8482641 0.82 DNMT1 (0.47) MAPTHTTTP53STAT3SMN1; SMN2
Triaziquone SCHEMBL8993238 0.82 DNMT1 (0.47) MAPTHTTTP53STAT3SMN1; SMN2
Triaziquone SCHEMBL6000230 0.82 DNMT1 (0.47) MAPTHTTTP53STAT3SMN1; SMN2
Triaziquone SCHEMBL7738777 0.82 DNMT1 (0.47) MAPTHTTTP53STAT3SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1019416-B1 LOW WATER POLYMERIC SILICONE COMPOSITIONS HAVING REDUCED MODULUS BAUSCH & LOMB (US) 2003-01-22 EP disclosed
EP-0865444-B1 MONOMERIC UNITS USEFUL FOR REDUCING THE MODULUS OF SILICONE HYDROGELS BAUSCH & LOMB (US) 2001-09-19 EP disclosed
EP-1019416-A1 MONOMERIC UNITS USEFUL FOR REDUCING THE MODULUS OF LOW WATER POLYMERIC SILICONE COMPOSITIONS BAUSCH & LOMB INCORPORATED (US) 2000-07-19 EP disclosed
US-5908906-A ESPECIALLY POLYMERS FROM 1-(3-METHACRYLOYLOXYPROPYL)-3-(1,1H-PERFLUOROPENTYLOXY)PROPYL) TETRAMETHYLDISILOXANE, CONTACT LENSES BAUSCH & LOMB INCORPORATED (US) 1999-06-01 US disclosed
EP-0865444-A1 MONOMERIC UNITS USEFUL FOR REDUCING THE MODULUS OF SILICONE HYDROGELS BAUSCH & LOMB INCORPORATED (US) 1998-09-23 EP disclosed
US-5714557-A UNSATURATED FLUORINATED ACRYLIC ESTER- OR AMIDE-CAPPED POLYSILOXANES AND DISILOXANES; CONTACT LENSES; FILMS; YOUNG'S MODULUS OF ELASTICIY; NONHYDROLYZING; MEDICAL EQUIPMENT BAUSCH & LOMB INCORPORATED (US) 1998-02-03 US disclosed
US-5710302-A Monomeric units useful for reducing the modules of silicone hydrogels BAUSCH & LOMB INCORPORATED (US) 1998-01-20 US disclosed
EP-0683799-B1 FLUOROSILICONE HYDROGELS BAUSCH & LOMB (US) 1997-12-29 EP disclosed
WO-1997020852-A1 MONOMERIC UNITS USEFUL FOR REDUCING THE MODULUS OF SILICONE HYDROGELS BAUSCH & LOMB INCORPORATED (US) 1997-06-12 WO disclosed
WO-1997020851-A1 MONOMERIC UNITS USEFUL FOR REDUCING THE MODULUS OF LOW WATER POLYMERIC SILICONE COMPOSITIONS BAUSCH & LOMB INCORPORATED (US) 1997-06-12 WO disclosed
US-5539016-A POLYMERS FOR CONTACT LENSES BAUSCH & LOMB INCORPORATED (US) 1996-07-23 US disclosed
EP-0683799-A1 FLUOROSILICONE HYDROGELS BAUSCH & LOMB INCORPORATED (US) 1995-11-29 EP disclosed
US-5387662-A For contact lenses; acrylated polysiloxanes BAUSCH & LOMB INCORPORATED (US) 1995-02-07 US disclosed
WO-1994018253-A1 FLUOROSILICONE HYDROGELS BAUSCH & LOMB INCORPORATED (US) 1994-08-18 WO disclosed
US-5321108-A Improving solubility of unsaturated siloxane monomers in hydrophilic monomer BAUSCH & LOMB INCORPORATED (US) 1994-06-14 US disclosed
EP-0340637-A2 Polymerization initiators WACKER-CHEMIE GMBH (DE) 1989-11-08 EP disclosed