SCHEMBL7017824

SCHEMBL7017824

CCn1c(=O)c2[nH]c(C)nc2n(C)c1=O

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 1/20 0.58
PDE1A P54750 1/20 0.58
PDE1B Q01064 1/20 0.58
PDE1C Q14123 1/20 0.58
ADORA2B P29275 4/20 0.56
ADORA2A P29274 3/20 0.55
PDE4A P27815 1/20 0.55
PDE4B Q07343 1/20 0.55
PDE4C Q08493 1/20 0.55
PDE4D Q08499 1/20 0.55
SIRT2 Q8IXJ6 1/20 0.51
SIRT1 Q96EB6 1/20 0.51
SIRT3 Q9NTG7 1/20 0.51
SIRT5 Q9NXA8 1/20 0.51
MAPK1 P28482 2/20 0.49
MEN1 O00255 1/20 0.49
LMNA P02545 1/20 0.49
CYP1A1 P04798 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28143495 0.87 SIRT1 (0.67) PDE2APDE1APDE1BPDE1CADORA2B
SCHEMBL27569373 0.86 PDE2A (0.57) PDE2APDE1APDE1BPDE1CADORA2B
SCHEMBL27598870 0.84 PDE2A (0.52) PDE2APDE1APDE1BPDE1CADORA2B
SCHEMBL20432543 0.83 PDE2A (0.55) PDE2APDE1APDE1BPDE1CADORA2B
SCHEMBL11072524 0.83 SIRT1 (0.55) PDE2APDE1APDE1BPDE1CADORA2B
SCHEMBL3949936 0.82 ADORA2B (0.59) PDE2APDE1APDE1BPDE1CADORA2B
SCHEMBL11066305 0.82 SIRT1 (0.54) PDE2APDE1APDE1BPDE1CADORA2B
SCHEMBL17609816 0.82 PDE2A (0.53) PDE2APDE1APDE1BPDE1CADORA2B
SCHEMBL18834910 0.82 PDE2A (0.53) PDE2APDE1APDE1BPDE1CADORA2B
SCHEMBL461786 0.81 PDE2A (0.62) PDE2APDE1APDE1BPDE1CADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998033382-A1 FUNGICIDAL COMPOSITIONS E.I. DU PONT DE NEMOURS AND COMPANY (US) 1998-08-06 WO claimed
WO-1998023155-A1 ARTHROPODICIDAL AND FUNGICIDAL CYCLIC AMIDES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1998-06-04 WO claimed
EP-0836384-A1 ARTHROPODICIDAL AND FUNGICIDAL CYCLIC AMIDES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1998-04-22 EP claimed
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
WO-1998033382-A1 FUNGICIDAL COMPOSITIONS E.I. DU PONT DE NEMOURS AND COMPANY (US) 1998-08-06 WO disclosed
US-5753664-A ANTITUMOR AGENTS, PYRIMIDONES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-05-19 US disclosed
EP-0836384-A1 ARTHROPODICIDAL AND FUNGICIDAL CYCLIC AMIDES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1998-04-22 EP disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed