SCHEMBL7019046

SCHEMBL7019046

CC(=O)C(=Cc1cc(Cl)c(S(C)(=O)=O)c(Cl)c1)C(C)=O

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.42
ALDH1A1 P00352 2/20 0.42
TDP1 Q9NUW8 2/20 0.40
GLA P06280 1/20 0.40
POLB P06746 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
GAA P10253 1/20 0.39
GPR35 Q9HC97 1/20 0.39
MAPT P10636 2/20 0.37
GLO1 Q04760 1/20 0.36
PTGS2 P35354 1/20 0.36
CA1 P00915 2/20 0.35
CA2 P00918 2/20 0.35
CA4 P22748 2/20 0.35
CA7 P43166 2/20 0.35
AKR1C3 P42330 5/20 0.34
AKR1C2 P52895 2/20 0.34
AKR1C1 Q04828 2/20 0.34
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7016901 0.79 TDP1 (0.46) KDM4EALDH1A1TDP1GLAPOLB
SCHEMBL7014950 0.76 TDP1 (0.46) KDM4EALDH1A1TDP1GLAPOLB
SCHEMBL7278497 0.74 GPR35 (0.58) KDM4EALDH1A1TDP1GLAPOLB
SCHEMBL5750483 0.74 KDM4E (0.50) KDM4EALDH1A1TDP1GLAPOLB
SCHEMBL7025723 0.74 ALDH1A1 (0.45) ALDH1A1TDP1L3MBTL1PTGS2LMNA
SCHEMBL7756019 0.73 ALDH1A1 (0.55) KDM4EALDH1A1TDP1GLAPOLB
Orazipone SCHEMBL1649524 0.69 ALDH1A1 (0.60) KDM4EALDH1A1TDP1GLAPOLB
SCHEMBL13271939 0.68 CA1 (0.41) ALDH1A1PTGS2CA1CA2LMNA
SCHEMBL7288527 0.66 ALDH1A1 (0.54) KDM4EALDH1A1TDP1L3MBTL1GAA
SCHEMBL10351283 0.66 ALDH1A1 (0.67) KDM4EALDH1A1TDP1GLAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1091933-B1 SUBSTITUTED BETA-DIKETONES AND THEIR USE ORION CORP (FI) 2003-11-26 EP claimed
EP-1091933-A1 SUBSTITUTED $g(b)-DIKETONES AND THEIR USE ORION CORPORATION (FI) 2001-04-18 EP claimed
US-6201027-B1 NONSTEROIDAL ANTIINFLAMMATORY DRUG FOR PROPHYLAXIS AND TREATMENT OF RESPIRATORY SYSTEM DISORDERS, I.E. ASTHMA, IN STEROID-RESISTANT MAMMALS ORION CORPORATION (FI) 2001-03-13 US claimed
WO-2000001667-A1 SUBSTITUTED β-DIKETONES AND THEIR USE ORION CORPORATION (FI) 2000-01-13 WO claimed
EP-1091933-B1 SUBSTITUTED BETA-DIKETONES AND THEIR USE ORION CORP (FI) 2003-11-26 EP disclosed
EP-1091933-A1 SUBSTITUTED $g(b)-DIKETONES AND THEIR USE ORION CORPORATION (FI) 2001-04-18 EP disclosed
US-6201027-B1 NONSTEROIDAL ANTIINFLAMMATORY DRUG FOR PROPHYLAXIS AND TREATMENT OF RESPIRATORY SYSTEM DISORDERS, I.E. ASTHMA, IN STEROID-RESISTANT MAMMALS ORION CORPORATION (FI) 2001-03-13 US disclosed
WO-2000001667-A1 SUBSTITUTED β-DIKETONES AND THEIR USE ORION CORPORATION (FI) 2000-01-13 WO disclosed