SCHEMBL7019238

SCHEMBL7019238

CCCOc1nc(SC)nc2[nH]ccc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 3/20 0.40
MAPK1 P28482 2/20 0.40
ADORA2A P29274 3/20 0.39
ADORA3 P0DMS8 2/20 0.39
LMNA P02545 3/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
HTT P42858 2/20 0.38
TTBK1 Q5TCY1 1/20 0.36
TTBK2 Q6IQ55 1/20 0.36
MAPT P10636 3/20 0.34
PDK1 Q15118 2/20 0.34
CDK1 P06493 1/20 0.34
CCNB1 P14635 1/20 0.34
CCNA2 P20248 1/20 0.34
CDK2 P24941 1/20 0.34
CCNA1 P78396 1/20 0.34
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
RECQL P46063 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7016051 0.88 LRRK2 (0.42) L3MBTL1TTBK1TTBK2MAPTPDK1
SCHEMBL7015802 0.82 NEK1 (0.39) L3MBTL1ADORA2AADORA3HTTPDK1
SCHEMBL4016987 0.80 MAPT (0.39) L3MBTL1MAPK1ADORA2ALMNASMN1; SMN2
SCHEMBL14029857 0.72 ADORA2A (0.43) L3MBTL1ADORA2ALMNAMAPTPDK1
SCHEMBL7655789 0.70 DYRK1A (0.42) L3MBTL1ADORA2ALMNAMAPTPDK1
SCHEMBL161735 0.70 ADORA2A (0.39) L3MBTL1MAPK1ADORA2ALMNASMN1; SMN2
SCHEMBL2564796 0.70 ADORA2A (0.42) L3MBTL1ADORA2ALMNASMN1; SMN2HTT
SCHEMBL10012874 0.70 ADORA2A (0.39) L3MBTL1ADORA2ALMNASMN1; SMN2HTT
SCHEMBL7015801 0.69 TTK (0.37) ADORA2ASMN1; SMN2PDK1LRRK2ADORA1
SCHEMBL11835880 0.69 CYP1A2 (0.51) LMNASMN1; SMN2CDK2CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed