SCHEMBL7015801

SCHEMBL7015801

CSc1nc(OC(C)OC(C)=O)c2cc[nH]c2n1

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TTK P33981 1/20 0.37
PDK1 Q15118 4/20 0.34
PDK2 Q15119 1/20 0.32
PDK3 Q15120 1/20 0.32
PDK4 Q16654 1/20 0.32
ADORA2A P29274 1/20 0.32
ADORA1 P30542 1/20 0.32
JAK3 P52333 1/20 0.32
LRRK2 Q5S007 2/20 0.31
TSHR P16473 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
HSD17B10 Q99714 1/20 0.31
CXCR2 P25025 1/20 0.30
JAK2 O60674 1/20 0.30
PDPK1 O15530 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7015802 0.77 NEK1 (0.39) PDK1ADORA2AJAK3LRRK2JAK2
SCHEMBL4016987 0.75 MAPT (0.39) PDK1ADORA2AADORA1LRRK2SMN1; SMN2
SCHEMBL7016051 0.72 LRRK2 (0.42) PDK1LRRK2
SCHEMBL7019238 0.69 L3MBTL1 (0.40) PDK1ADORA2AADORA1LRRK2SMN1; SMN2
SCHEMBL14004647 0.69 ADORA2A (0.37) PDK1PDK2PDK3PDK4ADORA2A
SCHEMBL161735 0.69 ADORA2A (0.39) PDK1PDK2PDK3PDK4ADORA2A
SCHEMBL7019102 0.68 JAK3 (0.35) TTKADORA2AADORA1JAK3LRRK2
SCHEMBL14029857 0.67 ADORA2A (0.43) PDK1PDK2PDK3PDK4ADORA2A
SCHEMBL7655789 0.66 DYRK1A (0.42) PDK1PDK2PDK3PDK4ADORA2A
SCHEMBL2564796 0.66 ADORA2A (0.42) PDK1ADORA2AADORA1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed