SCHEMBL7015802

SCHEMBL7015802

CSc1nc(OCCOC(C)=O)c2cc[nH]c2n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NEK1 Q96PY6 1/20 0.39
TP53 P04637 1/20 0.37
THRB P10828 1/20 0.37
ALDH1A1 P00352 1/20 0.37
HTT P42858 1/20 0.37
PDK1 Q15118 3/20 0.37
NUDT1 P36639 1/20 0.36
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
P2RY12 Q9H244 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
LRRK2 Q5S007 4/20 0.35
ADORA3 P0DMS8 1/20 0.34
ADORA2A P29274 1/20 0.34
JAK2 O60674 3/20 0.34
JAK3 P52333 2/20 0.34
JAK1 P23458 1/20 0.34
TYK2 P29597 1/20 0.34
CDK8 P49336 1/20 0.33
PPARG P37231 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7019238 0.82 L3MBTL1 (0.40) TP53ALDH1A1HTTPDK1NUDT1
SCHEMBL7016051 0.79 LRRK2 (0.42) ALDH1A1PDK1NUDT1L3MBTL1LRRK2
SCHEMBL4016987 0.74 MAPT (0.39) ALDH1A1HTTPDK1L3MBTL1LRRK2
SCHEMBL7019103 0.69 ALDH1A1 (0.49) NEK1ALDH1A1HTTJAK2JAK3
SCHEMBL29080497 0.69 NEK1 (0.46) NEK1NUDT1LRRK2JAK2JAK3
SCHEMBL161735 0.68 ADORA2A (0.39) ALDH1A1PDK1L3MBTL1LRRK2ADORA2A
SCHEMBL14029857 0.66 ADORA2A (0.43) ALDH1A1PDK1L3MBTL1ADORA2ADYRK1A
SCHEMBL2564796 0.65 ADORA2A (0.42) ALDH1A1HTTPDK1L3MBTL1ADORA2A
SCHEMBL7655789 0.65 DYRK1A (0.42) ALDH1A1PDK1L3MBTL1ADORA2ADYRK1A
SCHEMBL11832800 0.64 CDK2 (0.39) PDK1LRRK2JAK2JAK3PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733633-B1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-05-28 EP disclosed
EP-0733633-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-09-25 EP disclosed