SCHEMBL7019334

SCHEMBL7019334

O=C1COC2CCN(C(=O)[CH]Cc3ccncc3)C12

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CTSS P25774 8/20 0.40
CTSK P43235 7/20 0.40
CTSV O60911 4/20 0.40
CTSL P07711 3/20 0.40
ITGB3 P05106 2/20 0.32
ITGA2B P08514 2/20 0.32
GRM5 P41594 1/20 0.32
KDM4E B2RXH2 2/20 0.32
ALDH1A1 P00352 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7016835 0.87 CTSS (0.41) CTSSCTSKCTSVCTSL
SCHEMBL7017633 0.86 CTSS (0.40) CTSSCTSKCTSVCTSLALDH1A1
SCHEMBL7016638 0.86 CTSS (0.40) CTSSCTSKCTSVCTSLALDH1A1
SCHEMBL7018439 0.86 CTSS (0.40) CTSSCTSKCTSVCTSLSMN1; SMN2
SCHEMBL7023387 0.86 CTSS (0.40) CTSSCTSKCTSVCTSLALDH1A1
SCHEMBL6801912 0.84 CTSS (0.36) CTSSCTSKCTSVCTSL
SCHEMBL6801202 0.81 CTSK (0.37) CTSSCTSKCTSVCTSL
SCHEMBL7017077 0.81 CTSS (0.38) CTSSCTSKCTSVCTSLKMT2A
SCHEMBL7019497 0.81 CTSS (0.40) CTSSCTSKCTSVCTSL
SCHEMBL7013235 0.81 CTSS (0.37) CTSSCTSKCTSVCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1362052-A1 INHIBITORS OF CRUZIPAIN AND OTHER CYSTEINE PROTEASES Amura Therapeutics Limited (GB) 2003-11-19 EP disclosed
WO-2002057270-A1 INHIBITORS OF CRUZIPAIN AND OTHER CYSTEINE PROTEASES AMURA THERAPEUTICS LIMITED (GB) 2002-07-25 WO disclosed