SCHEMBL7019472

SCHEMBL7019472

CC(c1ccccc1)c1cncc(C(=O)N2CCC(c3cc(CN)ccc3O)CC2)c1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 1/20 0.41
TPSAB1 Q15661 7/20 0.39
KCNH2 Q12809 3/20 0.39
CYP2C9 P11712 2/20 0.38
CYP2C19 P33261 2/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
EGLN1 Q9GZT9 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4404742 0.99 MGLL (0.40) MGLLTPSAB1KCNH2CYP2C9CYP2C19
SCHEMBL1380986 0.91 MGLL (0.39) MGLLTPSAB1KCNH2CYP2C9CYP2C19
SCHEMBL1381850 0.90 TPSAB1 (0.48) MGLLTPSAB1KCNH2CYP2C9CYP2C19
Hydrochloric Acid SCHEMBL4401939 0.90 MGLL (0.38) MGLLTPSAB1KCNH2CYP2C9CYP2C19
Hydrochloric Acid SCHEMBL4414526 0.90 TPSAB1 (0.48) MGLLTPSAB1KCNH2CYP2C9CYP2C19
Hydrochloric Acid SCHEMBL4404465 0.85 TPSAB1 (0.51) TPSAB1
SCHEMBL7025345 0.84 MGLL (0.43) MGLLTPSAB1EGLN1
Hydrochloric Acid SCHEMBL4395981 0.84 TPSAB1 (0.41) MGLLTPSAB1EGLN1
SCHEMBL7019473 0.83 TPSAB1 (0.41) TPSAB1KCNH2CYP2C9CYP2C19MEN1
Hydrochloric Acid SCHEMBL4403351 0.83 MGLL (0.42) MGLLTPSAB1EGLN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1296972-A1 ARYLMETHYLAMINE DERIVATIVES FOR USE AS TRYPTASE INHIBITORS Aventis Pharmaceuticals Inc. (US) 2003-04-02 EP disclosed
WO-2001090101-A1 ARYLMETHYLAMINE DERIVATIVES FOR USE AS TRYPTASE INHIBITORS AVENTIS PHARMACEUTICALS INC. (US) 2001-11-29 WO disclosed