SCHEMBL7019991

SCHEMBL7019991

FC(F)(F)Oc1[c]cccc1-c1ccccc1Cl

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.34
DPP4 P27487 1/20 0.33
GPBAR1 Q8TDU6 1/20 0.33
HSD11B1 P28845 1/20 0.32
PDK2 Q15119 3/20 0.32
AR P10275 1/20 0.31
PIM1 P11309 1/20 0.31
CSNK2A2 P19784 1/20 0.31
CSNK2B P67870 1/20 0.31
PIM3 Q86V86 1/20 0.31
PIM2 Q9P1W9 1/20 0.31
GPR3 P46089 1/20 0.31
PTPRC P08575 1/20 0.31
NPC1 O15118 1/20 0.31
TP53 P04637 1/20 0.31
HPGD P15428 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
CHRM5 P08912 1/20 0.30
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL592798 0.84 GRIA1 (0.31) TDP1
SCHEMBL3540081 0.81 METAP2 (0.37) CYP2A6GPR3HPGD
SCHEMBL28839453 0.80 SLC6A4 (0.34) HSD11B1PDK2TP53SMN1; SMN2POLB
SCHEMBL3289120 0.80 HSD11B1 (0.41) HSD11B1ARHPGDTDP1
SCHEMBL5117336 0.78 NOTUM (0.41) HSD11B1PDK2
SCHEMBL9453855 0.77 CYP2A6 (0.38) CYP2A6DPP4HSD11B1PTPRCNPC1
SCHEMBL3971470 0.75 NOTUM (0.39) GPR3NPC1RAB9A
SCHEMBL3583635 0.74 CYP2A6 (0.38) CYP2A6DPP4GPBAR1HSD11B1PDK2
SCHEMBL15637646 0.73 PDK2 (0.35) PDK2
SCHEMBL6259560 0.73 ABL1 (0.38) PDK2RAB9APOLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1343768-A1 ARYL AND AMINOARYL SUBSTITUTED SEROTONIN RECEPTOR AGONIST AND ANTAGONIST LIGANDS Bristol-Myers Squibb Pharma Company (US) 2003-09-17 EP claimed
WO-2002059082-A2 ARYL AND AMINOARYL SUBSTITUTED SEROTONIN RECEPTOR AGONIST AND ANTAGONIST LIGANDS BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2002-08-01 WO claimed
EP-2903440-A1 HETEROCYCLIC COMPOUNDS AS PESTICIDES Bayer CropScience AG (DE) 2015-08-12 EP disclosed
WO-2014053450-A1 HETEROCYCLIC COMPOUNDS AS PESTICIDES BAYER CROPSCIENCE AG (DE) 2014-04-10 WO disclosed