SCHEMBL3971470

SCHEMBL3971470

FC(F)(F)Oc1ccc(-c2ccc[c]c2OC(F)(F)F)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.39
GPR3 P46089 2/20 0.38
FFAR4 Q5NUL3 2/20 0.38
FFAR1 O14842 1/20 0.38
KIF11 P52732 1/20 0.37
NISCH Q9Y2I1 1/20 0.37
SCN5A Q14524 4/20 0.37
SERPINE1 P05121 2/20 0.36
PRKDC P78527 1/20 0.35
KIT P10721 1/20 0.35
KDR P35968 1/20 0.35
FLT3 P36888 1/20 0.35
MAPT P10636 2/20 0.35
EPHX2 P34913 1/20 0.35
AURKA O14965 1/20 0.35
TPX2 Q9ULW0 1/20 0.35
KDM4E B2RXH2 1/20 0.35
NPC1 O15118 1/20 0.35
ALDH1A1 P00352 1/20 0.35
GAA P10253 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3540081 0.86 METAP2 (0.37) GPR3FFAR4FFAR1KIF11MAPT
SCHEMBL6259560 0.85 ABL1 (0.38) FFAR4FFAR1KIF11AURKATPX2
SCHEMBL28839453 0.85 SLC6A4 (0.34) FFAR4MAPTKDM4EALDH1A1
SCHEMBL6190102 0.82 ADORA1 (0.42) GPR3
SCHEMBL6573031 0.81 FFAR4 (0.40) NOTUMGPR3FFAR4FFAR1KIF11
SCHEMBL17840231 0.79 GPR3 (0.50) NOTUMGPR3FFAR4FFAR1KIF11
SCHEMBL4280164 0.76 PDK2 (0.45)
SCHEMBL3289120 0.75 HSD11B1 (0.41) NOTUMALDH1A1
SCHEMBL7019991 0.75 CYP2A6 (0.34) GPR3NPC1RAB9A
SCHEMBL15637646 0.75 PDK2 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7517901-B2 p38 MAP kinase inhibitors and methods for using the same ROCHE PALO ALTO LLC (US) 2009-04-14 US claimed
EP-1919877-A1 P38 MAP KINASE INHIBITORS AND METHODS FOR USING THE SAME F.HOFFMANN-LA ROCHE AG (CH) 2008-05-14 EP disclosed
WO-2007023114-A1 P38 MAP KINASE INHIBITORS AND METHODS FOR USING THE SAME F. HOFFMANN-LA ROCHE AG (CH) 2007-03-01 WO disclosed