SCHEMBL7020775

SCHEMBL7020775

COC(=O)[C@@H]1C[C@H](Oc2ccc(OC)cc2)CN1C(=O)OCc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
MMP9 P14780 4/20 0.47
MMP1 P03956 3/20 0.47
MMP3 P08254 3/20 0.47
MMP7 P09237 2/20 0.47
TP53 P04637 1/20 0.47
MMP13 P45452 1/20 0.47
POLB P06746 1/20 0.45
ADAM17 P78536 1/20 0.44
ADAM9 Q13443 1/20 0.44
MMP2 P08253 1/20 0.44
MMP8 P22894 1/20 0.44
KDM4E B2RXH2 1/20 0.43
LMNA P02545 1/20 0.43
PDE4B Q07343 1/20 0.42
MCL1 Q07820 2/20 0.42
FABP7 O15540 1/20 0.42
FABP5 Q01469 1/20 0.42
P2RX4 Q99571 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7020805 1.00 ALDH1A1 (0.48) ALDH1A1NPSR1MMP9MMP1MMP3
SCHEMBL7015458 0.95 POLB (0.47) ALDH1A1NPSR1TP53POLBKDM4E
SCHEMBL2298566 0.95 POLB (0.47) ALDH1A1NPSR1TP53POLBKDM4E
SCHEMBL7015459 0.95 POLB (0.47) ALDH1A1NPSR1TP53POLBKDM4E
SCHEMBL8999682 0.91 POLB (0.43) ALDH1A1NPSR1TP53POLBKDM4E
SCHEMBL7021955 0.90 MCL1 (0.45) ALDH1A1NPSR1TP53POLBKDM4E
SCHEMBL7021952 0.90 MCL1 (0.45) ALDH1A1NPSR1TP53POLBKDM4E
SCHEMBL8999667 0.89 HRH3 (0.43) ALDH1A1NPSR1TP53POLBKDM4E
SCHEMBL8999670 0.89 HRH3 (0.43) ALDH1A1NPSR1TP53POLBKDM4E
SCHEMBL7387119 0.89 POLB (0.45) ALDH1A1NPSR1MMP9MMP1MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1115704-B1 NOVEL SUBSTITUTED INDOLINONES WITH AN INHIBITORY EFFECT ON VARIOUS KINASES AND CYCLIN/CDK COMPLEXES BOEHRINGER INGELHEIM PHARMA (DE) 2003-06-18 EP disclosed
US-5693633-A Angiotensin II antagonists ELI LILLY AND COMPANY (US) 1997-12-02 US disclosed