SCHEMBL7023604

SCHEMBL7023604

COc1ccc(Cc2nnc([S+]([O-])CCC=C(F)F)o2)cc1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 1/20 0.44
ALDH1A1 P00352 12/20 0.41
TSHR P16473 6/20 0.41
LMNA P02545 4/20 0.41
HTT P42858 3/20 0.41
HPGD P15428 4/20 0.39
MAPT P10636 2/20 0.39
NCOA1 Q15788 1/20 0.39
NCOA3 Q9Y6Q9 1/20 0.39
PTK2 Q05397 1/20 0.39
KDM4E B2RXH2 1/20 0.38
HSD17B10 Q99714 1/20 0.38
POLB P06746 2/20 0.37
GAA P10253 1/20 0.36
TDP1 Q9NUW8 1/20 0.35
USP2 O75604 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7024884 0.82 NPC1 (0.46) RAB9AALDH1A1HTTHPGDMAPT
SCHEMBL7022967 0.73
SCHEMBL7020002 0.73 RAB9A (0.44) RAB9AALDH1A1TSHRLMNAHTT
SCHEMBL7021754 0.67 NPC1 (0.47) RAB9AALDH1A1TSHRHPGDMAPT
SCHEMBL10049321 0.66 CALM1 (0.50) ALDH1A1TSHRMAPT
SCHEMBL6053473 0.64 CALM1 (0.56) POLB
SCHEMBL7019727 0.63 MAPT (0.44) RAB9AALDH1A1MAPT
SCHEMBL10049317 0.63 ALDH1A1 (0.57) ALDH1A1TSHRHTT
SCHEMBL22577116 0.62
SCHEMBL22583884 0.62

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0749433-B1 (4,4-DIFLUOROBUT-3-ENYLTHIO)-SUBSTITUTED HETEROCYCLIC OR CARBOCYCLIC RING COMPOUNDS HAVING PESTICIDAL ACTIVITY SYNGENTA LTD (GB) 2003-05-07 EP disclosed
US-5952359-A NEMATICIDES, INSECTICIDES AND MITICIDES; 1,1-DIFLUORO-3-(THIAZOLYL OR ISOTHIAZOYL-THIO (OR SULFINYL OR SULFONYL)-PROP-1-ENE DERIVATIVES ZENECA LIMITED (GB) 1999-09-14 US disclosed
US-5912243-A NOVEL COMPOUNDS FOR CONTROLLING NEMATODES, INSECT OR ACARID PESTS ZENECA LIMITED (GB) 1999-06-15 US disclosed
US-5705516-A NEMATOCIDES, INSECTICIDES, ACARICIDES ZENECA LIMITED (GB) 1998-01-06 US disclosed
EP-0749433-A1 (4,4-DIFLUOROBUT-3-ENYLTHIO)-SUBSTITUTED HETEROCYCLIC OR CARBOCYCLIC RING COMPOUNDS HAVING PESTICIDAL ACTIVITY ZENECA LIMITED (GB) 1996-12-27 EP disclosed
WO-1995024403-A1 (4,4-DIFLUOROBUT-3-ENYLTHIO)-SUBSTITUTED HETEROCYCLIC OR CARBOCYCLIC RING COMPOUNDS HAVING PESTICIDAL ACTIVITY ZENECA LIMITED (GB) 1995-09-14 WO disclosed