SCHEMBL7025166

SCHEMBL7025166

CN1CCN(c2cccc3c2CC[C@@H](NC(=O)c2cccc(Oc4ccccc4)c2)C3)CC1

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.56
PKM P14618 1/20 0.54
DRD4 P21917 6/20 0.48
DRD2 P14416 3/20 0.48
ALDH1A1 P00352 1/20 0.48
GAA P10253 1/20 0.48
TSHR P16473 1/20 0.48
MTNR1A P48039 1/20 0.48
MTNR1B P49286 1/20 0.48
KMT2A Q03164 2/20 0.47
CCR3 P51677 1/20 0.45
MEN1 O00255 1/20 0.45
MAPT P10636 1/20 0.45
MCHR1 Q99705 1/20 0.44
KCNH2 Q12809 2/20 0.44
SCN9A Q15858 2/20 0.44
SCN5A Q14524 1/20 0.44
USP30 Q70CQ3 2/20 0.44
LMNA P02545 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7024171 1.00 NPC1 (0.56) NPC1PKMDRD4DRD2ALDH1A1
SCHEMBL7024175 1.00 NPC1 (0.56) NPC1PKMDRD4DRD2ALDH1A1
SCHEMBL7023936 0.93 NPC1 (0.56) NPC1PKMDRD4DRD2ALDH1A1
SCHEMBL7023930 0.93 NPC1 (0.56) NPC1PKMDRD4DRD2ALDH1A1
SCHEMBL7027929 0.81 MTNR1A (0.65) NPC1DRD4DRD2MTNR1AMTNR1B
SCHEMBL7027930 0.81 MTNR1A (0.65) NPC1DRD4DRD2MTNR1AMTNR1B
SCHEMBL4787207 0.80 MTNR1A (0.55) DRD4DRD2ALDH1A1GAATSHR
SCHEMBL7026958 0.80 MTNR1A (0.48) DRD4DRD2ALDH1A1GAATSHR
SCHEMBL7026953 0.80 MTNR1A (0.48) DRD4DRD2ALDH1A1GAATSHR
SCHEMBL7026344 0.77 MTNR1A (0.52) DRD4DRD2ALDH1A1GAATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0888319-B1 SUBSTITUTED 1,2,3,4-TETRAHYDRONAPHTHALENE DERIVATIVES ASTRAZENECA AB (SE) 2003-01-29 EP disclosed
US-6410530-B1 CENTRAL NERVOUS SYSTEM DISORDERS; PSYCHOLOGICAL DISORDERS ASTRAZENECA AB (SE) 2002-06-25 US disclosed
US-6124283-A Substituted 1,2,3,4-tetrahydronaphthalene derivatives ASTRA AKTIEBOLAG (SE) 2000-09-26 US disclosed