SCHEMBL7025675

SCHEMBL7025675

C=CC(CN)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.38
TDO2 P48775 1/20 0.38
IDO2 Q6ZQW0 1/20 0.38
PNMT P11086 2/20 0.37
TAAR1 Q96RJ0 1/20 0.37
AHR P35869 1/20 0.37
CYP3A4 P08684 5/20 0.35
SLC6A2 P23975 5/20 0.35
SLC6A4 P31645 5/20 0.35
SLC6A3 Q01959 5/20 0.35
CYP2D6 P10635 4/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
TSHR P16473 1/20 0.34
KCNH2 Q12809 2/20 0.33
TNF P01375 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13965635 0.81 SLC6A4 (0.38) IDO1TDO2IDO2AHRCYP3A4
SCHEMBL6006323 0.76 FFAR1 (0.46) ALDH1A1LMNAHTTSMN1; SMN2
SCHEMBL8332281 0.75 SLC6A3 (0.40) IDO1TDO2IDO2PNMTTAAR1
SCHEMBL8101480 0.75 SLC6A3 (0.40) IDO1TDO2IDO2PNMTTAAR1
SCHEMBL9618278 0.75 AHR (0.41) IDO1TDO2IDO2PNMTTAAR1
SCHEMBL18459577 0.75 IDO1 (0.39) IDO1TAAR1ALDH1A1HTTSMN1; SMN2
SCHEMBL16961922 0.74 AHR (0.44) IDO1TDO2IDO2AHRCYP3A4
SCHEMBL11078316 0.74 IDO1 (0.47) IDO1TDO2IDO2PNMTTAAR1
SCHEMBL1587058 0.72 PNMT (0.42) IDO1TDO2IDO2PNMTTAAR1
SCHEMBL12824482 0.71 CYP3A4 (0.43) IDO1TDO2IDO2PNMTTAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0934271-B1 SUBSTITUTED ARYLALKYLAMINES AS NEUROKININ ANTAGONISTS SCHERING CORP (US) 2003-09-03 EP disclosed
EP-0934271-A1 SUBSTITUTED ARYLALKYLAMINES AS NEUROKININ ANTAGONISTS SCHERING CORPORATION (US) 1999-08-11 EP disclosed
US-5789422-A PIPERIDINYL COMPOUNDS, TREATMENT OF ASTHMA, COUGH, MIGRAINE, CROHN*S DISEASE, ANTIINFLAMMATORY AGENTS SCHERING CORPORATION (US) 1998-08-04 US disclosed
WO-1998018761-A1 SUBSTITUTED ARYLALKYLAMINES AS NEUROKININ ANTAGONISTS SCHERING CORPORATION (US) 1998-05-07 WO disclosed