SCHEMBL7027900

SCHEMBL7027900

CN1CCN(c2cccc3c2C[C@H](NC(=O)c2csc(-c4ccncc4)n2)CC3)CC1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 5/20 0.48
CDK5 Q00535 2/20 0.48
CDK5R1 Q15078 2/20 0.48
ACKR3 P25106 4/20 0.46
IRAK4 Q9NWZ3 2/20 0.46
HPGD P15428 1/20 0.44
ROCK2 O75116 3/20 0.43
HTR3E A5X5Y0 1/20 0.42
HTR3B O95264 1/20 0.42
CHRNA7 P36544 1/20 0.42
HTR3A P46098 1/20 0.42
HTR3D Q70Z44 1/20 0.42
HTR3C Q8WXA8 1/20 0.42
PIM1 P11309 1/20 0.41
PIM3 Q86V86 1/20 0.41
PIM2 Q9P1W9 1/20 0.41
HRH2 P25021 1/20 0.40
HRH1 P35367 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7027905 1.00 CHEK1 (0.48) CHEK1CDK5CDK5R1ACKR3IRAK4
SCHEMBL7026213 0.94 HTR3E (0.49) CHEK1ACKR3IRAK4HTR3EHTR3B
SCHEMBL7026219 0.94 HTR3E (0.49) CHEK1ACKR3IRAK4HTR3EHTR3B
SCHEMBL7027930 0.76 MTNR1A (0.65)
SCHEMBL7027929 0.76 MTNR1A (0.65)
SCHEMBL7031820 0.75 MTNR1A (0.62)
SCHEMBL7031816 0.75 MTNR1A (0.62)
SCHEMBL7031005 0.75 MTNR1A (0.57)
SCHEMBL7031008 0.75 MTNR1A (0.57)
SCHEMBL7030412 0.74 MTNR1A (0.54)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0888319-B1 SUBSTITUTED 1,2,3,4-TETRAHYDRONAPHTHALENE DERIVATIVES ASTRAZENECA AB (SE) 2003-01-29 EP disclosed
US-6410530-B1 CENTRAL NERVOUS SYSTEM DISORDERS; PSYCHOLOGICAL DISORDERS ASTRAZENECA AB (SE) 2002-06-25 US disclosed
US-6124283-A Substituted 1,2,3,4-tetrahydronaphthalene derivatives ASTRA AKTIEBOLAG (SE) 2000-09-26 US disclosed