SCHEMBL7028611

SCHEMBL7028611

CN1CCN(C(C=O)c2ccc(Cl)cc2Cl)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 3/20 0.42
LMNA P02545 3/20 0.41
TP53 P04637 2/20 0.41
TSHR P16473 2/20 0.41
ALOX15 P16050 1/20 0.41
ALDH1A1 P00352 4/20 0.41
HTT P42858 2/20 0.41
KDM4E B2RXH2 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
MAPT P10636 1/20 0.41
CHRM2 P08172 1/20 0.40
HTR1A P08908 1/20 0.40
ADRA2A P08913 1/20 0.40
BCL2 P10415 1/20 0.40
CHRM1 P11229 1/20 0.40
DRD1 P21728 1/20 0.40
TBXA2R P21731 1/20 0.40
SLC6A2 P23975 1/20 0.40
SLC6A4 P31645 1/20 0.40
ADRA1A P35348 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7019221 0.82 CNR1 (0.47) LMNATP53ALDH1A1HTTKDM4E
SCHEMBL14968308 0.72 ESR1 (0.45) ALDH1A1SMN1; SMN2SLC6A2SLC6A4SLC6A3
SCHEMBL20772370 0.69 HSD17B2 (0.43) TDP1LMNATP53TSHRALOX15
SCHEMBL838659 0.69 TP53 (0.57) TDP1LMNATP53HTTSMN1; SMN2
SCHEMBL12066465 0.68 CHRM1 (0.59) TDP1LMNATSHRALDH1A1KDM4E
SCHEMBL13258519 0.68 CHRM1 (0.59) TDP1LMNATSHRALDH1A1KDM4E
SCHEMBL20775033 0.68 ALDH1A1 (0.40) TSHRALDH1A1HTTKDM4ESMN1; SMN2
SCHEMBL7575571 0.68 TP53 (0.50) TDP1LMNATP53TSHRALDH1A1
SCHEMBL7021943 0.67 LMNA (0.41) TDP1LMNATP53TSHRALOX15
SCHEMBL10805341 0.67 CYP19A1 (0.50) TDP1LMNATP53TSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1317433-A2 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 2003-06-11 EP disclosed
WO-2002020495-A2 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 2002-03-14 WO disclosed
EP-1087963-A1 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 Chiron Corporation (US) 2001-04-04 EP disclosed
WO-1999065897-A1 INHIBITORS OF GLYCOGEN SYNTHASE KINASE 3 CHIRON CORPORATION (US) 1999-12-23 WO disclosed