SCHEMBL7030337

SCHEMBL7030337

N#Cc1ccc(C#CCCO)cc1.N#Cc1ccc(CCCCO)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.46
HSD17B10 Q99714 1/20 0.46
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
FFAR1 O14842 4/20 0.40
FFAR4 Q5NUL3 2/20 0.40
KCNJ1 P48048 1/20 0.39
KCNH2 Q12809 1/20 0.39
CA2 P00918 2/20 0.38
HRH3 Q9Y5N1 1/20 0.38
LOXL2 Q9Y4K0 2/20 0.38
CYP2A6 P11509 1/20 0.38
CYP19A1 P11511 1/20 0.36
CYP4F2 P78329 1/20 0.36
CYP4A11 Q02928 1/20 0.36
GABRP O00591 1/20 0.35
GABRD O14764 1/20 0.35
GABRA1 P14867 1/20 0.35
GABRB1 P18505 1/20 0.35
GABRG2 P18507 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2959480 0.87 TSHR (0.58) TSHRHSD17B10CYP11B1CYP11B2KCNJ1
SCHEMBL7396265 0.85 TSHR (0.61) TSHRHSD17B10CYP11B1CYP11B2KCNJ1
SCHEMBL4060135 0.85 TSHR (0.61) TSHRHSD17B10CYP11B1CYP11B2KCNJ1
SCHEMBL5631364 0.85 CA2 (0.44) TSHRCA2HRH3LOXL2CYP2A6
SCHEMBL21623419 0.83 TSHR (0.56) TSHRHSD17B10FFAR1FFAR4KCNJ1
SCHEMBL21623468 0.83 TSHR (0.50) TSHRHSD17B10FFAR1FFAR4KCNJ1
SCHEMBL7395296 0.81 GABRP (0.47) CYP11B1CYP11B2FFAR1FFAR4CA2
SCHEMBL81846 0.81 TSHR (0.55) TSHRHSD17B10CYP11B1CYP11B2KCNJ1
SCHEMBL10569888 0.77 TSHR (0.68) TSHRHSD17B10KCNJ1KCNH2CA2
SCHEMBL10773059 0.76 TSHR (0.64) TSHRHSD17B10CYP11B1CYP11B2KCNJ1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1389211-A1 3,7-DIAZYBICYCLO 3.3.1] FORMULATIONS AS ANTIARRHYTMIC COMPOUNDS AstraZeneca AB (SE) 2004-02-18 EP disclosed
WO-2002083687-A1 3,7-DIAZYBICYCLO [3.3.1] FORMULATIONS AS ANTIARRHYTMIC COMPOUNDS ASTRAZENECA AB (SE) 2002-10-24 WO disclosed