SCHEMBL7030552

SCHEMBL7030552

O=c1[nH]c(=O)c2cc(Cc3ccc[nH]3)ccc2[nH]1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.44
KDM4E B2RXH2 3/20 0.44
CA12 O43570 2/20 0.44
CA9 Q16790 2/20 0.44
PDE3A Q14432 1/20 0.36
GAA P10253 1/20 0.36
PKM P14618 1/20 0.36
TYMP P19971 1/20 0.36
GSK3B P49841 1/20 0.36
BACE1 P56817 1/20 0.36
HPGD P15428 3/20 0.36
ALDH1A1 P00352 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
SIRT6 Q8N6T7 2/20 0.35
SIRT2 Q8IXJ6 1/20 0.35
PARG Q86W56 1/20 0.35
MEN1 O00255 1/20 0.33
MAPT P10636 1/20 0.33
KMT2A Q03164 1/20 0.33
HSD17B10 Q99714 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7028533 0.79 KDM4E (0.53) PARP1KDM4ECA12CA9PDE3A
SCHEMBL7025839 0.75 CA12 (0.45) PARP1KDM4ECA12CA9PDE3A
SCHEMBL2056368 0.73 ALDH1A1 (0.50) PARP1KDM4ECA12CA9GAA
SCHEMBL20942693 0.73 GAA (0.66) PARP1KDM4ECA12CA9PDE3A
SCHEMBL7028337 0.73 CA12 (0.50) PARP1KDM4ECA12CA9PDE3A
SCHEMBL7034143 0.73 CA12 (0.50) PARP1KDM4ECA12CA9PDE3A
SCHEMBL9761081 0.73 KDM4E (0.46) PARP1KDM4ECA12CA9GAA
SCHEMBL7029630 0.73 KDM4E (0.53) PARP1KDM4ECA12CA9PDE3A
SCHEMBL7028562 0.71 CA12 (0.47) PARP1KDM4ECA12CA9PDE3A
SCHEMBL7033620 0.71 CA12 (0.47) PARP1KDM4ECA12CA9GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0878468-B1 Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL CO (JP) 2003-03-19 EP disclosed
EP-0775697-B1 Process for producing 1-substituted tetrahydroquinazolindionen SUMITOMO CHEMICAL CO (JP) 2003-02-12 EP disclosed
US-5994542-A Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1999-11-30 US disclosed
EP-0878468-A1 Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1998-11-18 EP disclosed
US-5756738-A Process for producing 1-substituted tetrahydroquinazolines SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1998-05-26 US disclosed
EP-0775697-A1 Process for producing 1-substituted tetrahydroquinazolindionen SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1997-05-28 EP disclosed