SCHEMBL7032960

SCHEMBL7032960

COc1ccc2c(c1)C(C)(O)CC(C)(C)CO2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2B P41595 2/20 0.42
SIGMAR1 Q99720 2/20 0.42
HTR1A P08908 1/20 0.42
HTR7 P34969 1/20 0.41
TMEM97 Q5BJF2 1/20 0.41
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
CYP3A4 P08684 1/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
MAPK1 P28482 1/20 0.38
HSD17B10 Q99714 1/20 0.38
BACE1 P56817 11/20 0.36
KLK7 P49862 1/20 0.36
CTSD P07339 5/20 0.35
RARB P10826 1/20 0.35
RARG P13631 1/20 0.35
PDK2 Q15119 1/20 0.35
MEN1 O00255 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7028281 0.79 CTSD (0.42) HTR2BSIGMAR1HTR1AKDM4EALDH1A1
SCHEMBL11455838 0.78 HTR2B (0.48) HTR2BSIGMAR1HTR1AHTR7TMEM97
SCHEMBL8314935 0.77 SCN9A (0.38) HTR2BSIGMAR1HTR1AHTR7TMEM97
SCHEMBL9832996 0.76 HTR2B (0.46) HTR2BSIGMAR1HTR1AHTR7TMEM97
SCHEMBL8315522 0.75 BACE1 (0.33) HTR2BSIGMAR1HTR1AHTR7TMEM97
SCHEMBL14031240 0.74 TAAR1 (0.34)
SCHEMBL5734820 0.72 KMT2A (0.43) HTR2BSIGMAR1HTR1AALDH1A1MAPT
SCHEMBL31525286 0.72 HTR2B (0.43) HTR2BSIGMAR1HTR1AHTR7TMEM97
SCHEMBL3378398 0.71 KDM4E (0.45) HTR2BSIGMAR1HTR1AHTR7TMEM97
SCHEMBL9385665 0.70 HTR2B (0.44) HTR2BSIGMAR1HTR1AHTR7TMEM97

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6596758-B1 Treatment of dislipidaemias, atherosclerosis and diabetes, to pharmaceutical compositions comprising them and to processes allowing the preparation of these compounds. MERCK PATENT GMBH (DE) 2003-07-22 US disclosed
EP-1140893-B1 BENZOPYRANS AND BENZOXEPINES, PHARMACEUTICAL COMPOSITIONS COMPRISING THEM AND PREPARATION PROCESS MERCK PATENT GMBH (DE) 2003-03-05 EP disclosed