SCHEMBL8314935

SCHEMBL8314935

COc1ccc2c(c1)C(O)(c1ccccn1)CC(C)(C)CO2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.38
BACE1 P56817 7/20 0.36
CTSD P07339 5/20 0.36
HTR2B P41595 2/20 0.36
SIGMAR1 Q99720 2/20 0.36
HTR7 P34969 1/20 0.36
TMEM97 Q5BJF2 1/20 0.36
PDK2 Q15119 2/20 0.36
SLC6A2 P23975 1/20 0.35
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
GAA P10253 1/20 0.34
HTR1A P08908 1/20 0.34
RAB9A P51151 2/20 0.33
NPC1 O15118 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8311682 0.87 BACE1 (0.36) SCN9ABACE1CTSDPDK2SLC6A2
SCHEMBL8310494 0.85 SCN9A (0.38) SCN9ASLC6A2HTR1ARAB9ANPC1
SCHEMBL8316835 0.85 SLC6A2 (0.39) HTR2BSIGMAR1PDK2SLC6A2GAA
SCHEMBL8311266 0.85 SLC6A2 (0.37) BACE1PDK2SLC6A2
SCHEMBL8311974 0.84 BACE1 (0.37) BACE1SLC6A2KMT2AALDH1A1MAPT
SCHEMBL8313637 0.84 SLC6A2 (0.36) BACE1SLC6A2KMT2ARAB9ANPC1
SCHEMBL8310708 0.83 SLC6A2 (0.40) PDK2SLC6A2KMT2AHTR1ASMN1; SMN2
SCHEMBL8314119 0.83 HTR2B (0.38) BACE1CTSDHTR2BSIGMAR1HTR7
SCHEMBL8313766 0.82 PDK2 (0.35) PDK2SLC6A2
SCHEMBL8313905 0.82 PDK2 (0.35) BACE1PDK2SLC6A2KMT2ARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0626954-B1 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1999-03-17 EP disclosed
US-5602152-A POTASSIUM CHANNEL MODULATOR MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-02-11 US disclosed
WO-1994013658-A2 BENZOCYCLOHEPTENES, BENZOXEPINES AND BENZOTHIEPINES MERCK PATENT GMBH (DE) 1994-06-23 WO disclosed