SCHEMBL7036713

SCHEMBL7036713

O=Cc1cnc(C(c2ccccc2)(c2ccccc2)c2ccccc2)[nH]1

nearest known ligand 0.33

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.33
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19209069 0.73 MASP2 (0.32)
SCHEMBL9424713 0.70
SCHEMBL2293472 0.69 SCN2A (0.55)
SCHEMBL7255232 0.69 AOC3 (0.34) ALDH1A1
SCHEMBL7537360 0.67 ERN1 (0.33) ALDH1A1
SCHEMBL4439049 0.67 HPGDS (0.50)
SCHEMBL2488026 0.66 P2RX7 (0.32) CYP2A6ALDH1A1
SCHEMBL7819462 0.65 CYP19A1 (0.39) CYP2A6ALDH1A1
SCHEMBL15332010 0.63 SCN2A (0.65) ALDH1A1
SCHEMBL4028445 0.62 NPSR1 (0.61) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3400226-A1 DERIVATIVES OF PYRROLOIMIDAZOLE OR ANALOGUES THEREOF WHICH ARE USEFUL FOR THE TREATMENT OF INTER ALIA CANCER Emcure Pharmaceuticals Limited (IN) 2018-11-14 EP disclosed
WO-2017134555-A1 DERIVATIVES OF PYRROLOIMIDAZOLE OR ANALOGUES THEREOF WHICH ARE USEFUL FOR THE TREATMENT OF INTER ALIA CANCER EMCURE PHARMACEUTICALS LIMITED (IN) 2017-08-10 WO disclosed
WO-2003099812-A1 PHENYL-FURAN OR PHENYL-THIOPHENE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS MEDICINE PIERRE FABRE MEDICAMENT (FR) 2003-12-04 WO disclosed
WO-2003006012-A1 COMPOUNDS AND METHODS FOR THE INHIBITION OF TRYPANOSOMA CRUZ I YALE UNIVERSITY (US) 2003-01-23 WO disclosed