SCHEMBL7038368

SCHEMBL7038368

C=C(C)c1nn2ccccc2c1-c1ccc(=O)n(CCOC)n1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 1/20 0.48
KDM4E B2RXH2 3/20 0.36
ALDH1A1 P00352 2/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
HSD17B10 Q99714 1/20 0.35
PDE5A O76074 1/20 0.34
PDE3A Q14432 1/20 0.34
PTGDR2 Q9Y5Y4 2/20 0.34
POLB P06746 1/20 0.34
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
KDM4C Q9H3R0 1/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7036909 0.82 ADORA1 (0.43) ADORA1KDM4EALDH1A1MEN1KMT2A
SCHEMBL7035541 0.82 ADORA1 (0.45) ADORA1KDM4EPDE5APDE3APTGDR2
SCHEMBL7033867 0.81 ADORA1 (0.47) ADORA1KDM4EHSD17B10PDE5APDE3A
SCHEMBL7036654 0.81 ADORA1 (0.44) ADORA1ALDH1A1PDE5APDE3APTGDR2
SCHEMBL7035962 0.80 ADORA1 (0.43) ADORA1KDM4EALDH1A1PDE5APDE3A
SCHEMBL7039890 0.77 PDE5A (0.42) ADORA1ALDH1A1MEN1KMT2APDE5A
SCHEMBL7032871 0.72 PDE3A (0.65) ADORA1ALDH1A1MEN1KMT2APDE5A
SCHEMBL7033864 0.72 ADORA1 (0.38) ADORA1PDE5APDE3APDE4B
SCHEMBL8808083 0.71 ADORA1 (0.73) ADORA1KDM4EALDH1A1MEN1KMT2A
SCHEMBL8809084 0.71 ADORA1 (0.67) ADORA1KDM4EHSD17B10HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003004494-A1 PYRIDAZINONE COMPOUND AS ADENOSINE ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2003-01-16 WO disclosed