SCHEMBL7039253

SCHEMBL7039253

COc1ccc(C(C(=O)N(Cc2ccc(CNC(N)=O)cc2)[C@H](CCCNC(=N)N)C(=O)NCC(=O)O)c2ccc(OC)cc2)cc1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CASR P41180 1/20 0.38
KMT2A Q03164 4/20 0.37
CNR1 P21554 1/20 0.37
CNR2 P34972 1/20 0.37
ITGB3 P05106 2/20 0.36
ITGA2B P08514 2/20 0.36
ALDH1A1 P00352 3/20 0.36
TSHR P16473 1/20 0.36
HSD17B10 Q99714 1/20 0.36
MEN1 O00255 3/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
POLB P06746 1/20 0.35
YAP1 P46937 1/20 0.35
TEAD4 Q15561 1/20 0.35
GAA P10253 1/20 0.34
CXCR3 P49682 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7036782 0.92 EPOR (0.36) KMT2AITGB3ITGA2BMEN1
SCHEMBL7043493 0.91 MEN1 (0.35) KMT2AITGB3ITGA2BMEN1POLB
SCHEMBL6900020 0.91 CASR (0.38) CASRKMT2ACNR1CNR2ITGB3
SCHEMBL6901717 0.85 EPOR (0.35) ITGB3ITGA2BALDH1A1TSHR
SCHEMBL8526883 0.84 NPY1R (0.34) ITGB3ITGA2B
SCHEMBL8528634 0.83 NPY1R (0.37) KMT2AMEN1POLB
SCHEMBL9196992 0.83 CNR1 (0.42) CASRKMT2ACNR1CNR2ITGB3
SCHEMBL8121285 0.83 EPOR (0.41) KMT2AMEN1
SCHEMBL8526482 0.83 KMT2A (0.40) KMT2AITGB3ITGA2BALDH1A1TSHR
SCHEMBL9195083 0.83 CNR1 (0.43) CASRKMT2ACNR1CNR2ITGB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0885186-B1 AMINO ACID DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS AND PROCESSES FOR PREPARING THEM THOMAE GMBH DR K (DE) 2003-03-26 EP disclosed
EP-0885186-A1 AMINO ACID DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS AND PROCESSES FOR PREPARING THEM Dr. Karl Thomae GmbH (DE) 1998-12-23 EP disclosed
WO-1997019911-A1 AMINO ACID DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS AND PROCESSES FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1997-06-05 WO disclosed