SCHEMBL8526482

SCHEMBL8526482

COc1ccc2cc(C(=O)N(Cc3ccc(CNC(N)=O)cc3)[C@H](CCCNC(=N)N)C(=O)NCC(=O)O)ccc2c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
MCHR1 Q99705 1/20 0.39
ITGB3 P05106 3/20 0.36
ITGA2B P08514 3/20 0.36
ALDH1A1 P00352 3/20 0.36
HSD17B10 Q99714 2/20 0.36
CYP2C19 P33261 2/20 0.36
CYP1A2 P05177 1/20 0.36
HPGD P15428 1/20 0.36
PROC P04070 2/20 0.36
TSHR P16473 1/20 0.35
CXCR3 P49682 1/20 0.35
PRSS1 P07477 1/20 0.34
TMPRSS15 P98073 1/20 0.34
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
F2 P00734 2/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8528194 0.90 F7 (0.40) MCHR1PROCF2HDAC3HDAC1
SCHEMBL7039253 0.83 CASR (0.38) KMT2AMEN1ITGB3ITGA2BALDH1A1
SCHEMBL8526111 0.83 TMEM97 (0.38) ITGB3ITGA2BPROCF2
SCHEMBL8122129 0.82 F7 (0.40) PROCF2
SCHEMBL8526191 0.81 F7 (0.42) MCHR1F2HDAC3HDAC1HDAC2
SCHEMBL8528338 0.81 CCR2 (0.36) MCHR1F2
SCHEMBL8527067 0.79 ALDH1A1 (0.41) KMT2AMEN1MCHR1ALDH1A1HPGD
SCHEMBL7043493 0.77 MEN1 (0.35) KMT2AMEN1ITGB3ITGA2B
SCHEMBL7036782 0.77 EPOR (0.36) KMT2AMEN1ITGB3ITGA2B
SCHEMBL8121011 0.77 F7 (0.37) PROCSLC6A2SLC6A4F2HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0885186-A1 AMINO ACID DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS AND PROCESSES FOR PREPARING THEM Dr. Karl Thomae GmbH (DE) 1998-12-23 EP disclosed
WO-1997019911-A1 AMINO ACID DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS AND PROCESSES FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1997-06-05 WO disclosed